Drug_ID Target_name Uniprot_ID MOA ReferenceID DG00234 5-HT 1B receptor (HTR1B) 5HT1B_HUMAN Modulator REF00002872 DG01217 5-HT 1F receptor (HTR1F) 5HT1F_HUMAN Agonist REF00003758 DG01201 5-HT 2A receptor (HTR2A) 5HT2A_HUMAN Agonist REF00003307 DG01505 5-HT 2A receptor (HTR2A) 5HT2A_HUMAN Agonist REF00004318 DG00679 5-HT 3 receptor (5HT3R) NOUNIPROTAC Antagonist REF00003082 DG00640 5-HT 3A receptor (HTR3A) 5HT3A_HUMAN Blocker (channel blocker) REF00003593 DG01160 5-HT 3A receptor (HTR3A) 5HT3A_HUMAN Blocker (channel blocker) REF00003748 DG01315 5-HT 4 receptor (HTR4) 5HT4R_HUMAN Agonist REF00003459 DG00695 Acetylcholinesterase (AChE) ACES_HUMAN Inhibitor REF00003641 DG01463 Acetylcholinesterase (AChE) ACES_HUMAN Inhibitor REF00004328 DG00165 Acetyl-CoA carboxylase 2 (ACACB) ACACB_HUMAN Activator REF00002447 DG00052 Acetyl-CoA:lyso-PAF acetyltransferase (PCAT) PCAT1_HUMAN; PCAT2_HUMAN Inhibitor REF00002268 DG01822 Acetyl-CoA:lyso-PAF acetyltransferase (PCAT) PCAT1_HUMAN; PCAT2_HUMAN Inhibitor REF00003899 DG01320 Activation B7-1 antigen (CD80) CD80_HUMAN . REF00003131 DG01801 Adenosine A2b receptor (ADORA2B) AA2BR_HUMAN Agonist REF00004202 DG00179 Adenosine deaminase (ADA) ADA_HUMAN Inhibitor REF00001069 DG00883 Adenosine deaminase (ADA) ADA_HUMAN Inhibitor REF00003290 DG00775 Adrenergic receptor Alpha-1 (ADRA1) NOUNIPROTAC Antagonist REF00003134 DG00844 Adrenergic receptor alpha-1B (ADRA1B) ADA1B_HUMAN Antagonist REF00003706 DG00868 Adrenergic receptor alpha-1B (ADRA1B) ADA1B_HUMAN Antagonist REF00003643 DG00707 Adrenergic receptor Alpha-2 (ADRA2) NOUNIPROTAC Antagonist REF00003389 DG01153 Adrenergic receptor Alpha-2 (ADRA2) NOUNIPROTAC Antagonist REF00003642 DG00707 Adrenergic receptor alpha-2C (ADRA2C) ADA2C_HUMAN Modulator REF00003389 DG00988 Adrenergic receptor alpha-2C (ADRA2C) ADA2C_HUMAN Modulator REF00003649 DG00759 Adrenergic receptor beta-1 (ADRB1) ADRB1_HUMAN Antagonist REF00003160 DG00931 Adrenergic receptor beta-1 (ADRB1) ADRB1_HUMAN Antagonist REF00003603 DG00959 Adrenergic receptor beta-1 (ADRB1) ADRB1_HUMAN Antagonist REF00003247 DG01466 Adrenergic receptor beta-1 (ADRB1) ADRB1_HUMAN Antagonist REF00003942 DG00759 Adrenergic receptor beta-2 (ADRB2) ADRB2_HUMAN Agonist REF00003160 DG00923 Adrenergic receptor beta-2 (ADRB2) ADRB2_HUMAN Agonist REF00003713 DG01213 Adrenergic receptor beta-2 (ADRB2) ADRB2_HUMAN Agonist REF00003628 DG01466 Adrenergic receptor beta-2 (ADRB2) ADRB2_HUMAN Agonist REF00003942 DG01255 Adrenergic receptor beta-3 (ADRB3) ADRB3_HUMAN Agonist REF00003554 DG00103 Albendazole monooxygenase (CYP3A4) CP3A4_HUMAN Inhibitor REF00002220 DG00666 Albendazole monooxygenase (CYP3A4) CP3A4_HUMAN Inhibitor REF00003409 DG00006 Aldose reductase (AKR1B1) ALDR_HUMAN Inhibitor REF00002102 DG01074 Aldose reductase (AKR1B1) ALDR_HUMAN Modulator REF00003401 DG00050 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Modulator REF00002690 DG00053 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Inhibitor REF00002690 DG00056 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Modulator REF00001377 DG00270 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Inhibitor REF00001979 DG00630 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Inhibitor REF00003465 DG00632 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Inhibitor REF00003465 DG01520 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Inhibitor REF00004563 DG01605 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Inhibitor REF00004474 DG01618 ALK tyrosine kinase receptor (ALK) ALK_HUMAN Inhibitor REF00004504 DG00134 Amidophosphoribosyltransferase (PPAT) PUR1_HUMAN Breaker REF00001406 DG00614 Amidophosphoribosyltransferase (PPAT) PUR1_HUMAN Inhibitor REF00003094 DG00829 Amiloride-sensitive sodium channel (ENaC) SCNNA_HUMAN; SCNNB_HUMAN; SCNNG_HUMAN; SCNND_HUMAN Activator REF00003271 DG00103 Amyloid beta A4 protein (APP) A4_HUMAN Inhibitor REF00002220 DG00247 Androgen receptor (AR) ANDR_HUMAN Modulator REF00001776 DG00705 Androgen receptor (AR) ANDR_HUMAN Antagonist REF00002983 DG00861 Androgen receptor (AR) ANDR_HUMAN Antagonist REF00003187 DG00981 Androgen receptor (AR) ANDR_HUMAN Antagonist REF00003724 DG00006 Androgen receptor messenger RNA (AR mRNA) ANDR_HUMAN Inhibitor REF00002102 DG01004 Angiogenesis/myeloma cell growth (AMCG) NOUNIPROTAC Modulator REF00003511 DG00938 Angiotensin II receptor type-1 (AGTR1) AGTR1_HUMAN . REF00003325 DG01158 Angiotensin II receptor type-1 (AGTR1) AGTR1_HUMAN . REF00003482 DG01811 Angiotensin II receptor type-1 (AGTR1) AGTR1_HUMAN . REF00004204 DG01158 Angiotensin II receptor type-2 (AGTR2) AGTR2_HUMAN Antagonist REF00003482 DG01811 Angiotensin II receptor type-2 (AGTR2) AGTR2_HUMAN Antagonist REF00004204 DG00327 Angiotensin-converting enzyme (ACE) ACE_HUMAN Modulator REF00002541 DG01157 Angiotensinogenase renin (REN) RENI_HUMAN Inhibitor REF00003855 DG00151 Apoptosis regulator Bcl-2 (BCL-2) BCL2_HUMAN Modulator REF00002764 DG01268 Apoptosis regulator Bcl-2 (BCL-2) BCL2_HUMAN Modulator REF00003512 DG01586 Apoptosis regulator Bcl-2 (BCL-2) BCL2_HUMAN Modulator REF00001577 DG01824 Arachidonate 12-lipoxygenase (12-LOX) LOX12_HUMAN Inhibitor REF00003895 DG01824 Arachidonate 15-lipoxygenase (15-LOX) LOX15_HUMAN Inhibitor REF00003895 DG00010 Arachidonate 5-lipoxygenase (5-LOX) LOX5_HUMAN Inhibitor REF00002302 DG00402 Arachidonate 5-lipoxygenase (5-LOX) LOX5_HUMAN Inhibitor REF00000712 DG00725 Arachidonate 5-lipoxygenase (5-LOX) LOX5_HUMAN Modulator REF00003673 DG00006 Aromatase (CYP19A1) CP19A_HUMAN Inhibitor REF00002102 DG00397 Aromatase (CYP19A1) CP19A_HUMAN Inhibitor REF00001681 DG00403 Aromatase (CYP19A1) CP19A_HUMAN Inhibitor REF00001616 DG00422 Aromatase (CYP19A1) CP19A_HUMAN Inhibitor REF00001681 DG00343 Asparaginase (ASRGL1) ASGL1_HUMAN Modulator REF00001382 DG00915 ATP-binding cassette transporter C9 (ABCC9) ABCC9_HUMAN Blocker REF00003444 DG00039 ATP-binding cassette transporter G2 (ABCG2) ABCG2_HUMAN Inhibitor REF00002801 DG00068 Bacterial 16S ribosomal RNA (Bact 16S rRNA) . Binder REF00001005 DG00119 Bacterial 16S ribosomal RNA (Bact 16S rRNA) . Inhibitor REF00002517 DG00145 Bacterial 16S ribosomal RNA (Bact 16S rRNA) . Inhibitor REF00000654 DG00265 Bacterial 16S ribosomal RNA (Bact 16S rRNA) . Inhibitor REF00002824 DG00432 Bacterial 16S ribosomal RNA (Bact 16S rRNA) . Inhibitor REF00002873 DG01604 Bacterial 16S ribosomal RNA (Bact 16S rRNA) NOUNIPROTAC Inhibitor REF00004359 DG00106 Bacterial 23S ribosomal RNA (Bact 23S rRNA) . Binder REF00002431 DG00182 Bacterial 23S ribosomal RNA (Bact 23S rRNA) . Binder REF00000645 DG00188 Bacterial 23S ribosomal RNA (Bact 23S rRNA) . Binder REF00000654 DG00242 Bacterial 23S ribosomal RNA (Bact 23S rRNA) . Binder REF00000593 DG00272 Bacterial 23S ribosomal RNA (Bact 23S rRNA) . Modulator REF00001700 DG00293 Bacterial 23S ribosomal RNA (Bact 23S rRNA) . Binder REF00002294 DG00086 Bacterial 30S ribosomal RNA (Bact 30S rRNA) . Modulator REF00001622 DG00261 Bacterial 30S ribosomal RNA (Bact 30S rRNA) . Modulator REF00002431 DG00400 Bacterial 30S ribosomal RNA (Bact 30S rRNA) . Modulator REF00000775 DG01148 Bacterial 30S ribosomal RNA (Bact 30S rRNA) NOUNIPROTAC Inhibitor REF00003449 DG01465 Bacterial 30S ribosomal RNA (Bact 30S rRNA) NOUNIPROTAC Inhibitor REF00003941 DG00038 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Binder REF00000619 DG00043 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Modulator REF00000798 DG00063 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Binder REF00001049 DG00127 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Binder REF00000619 DG00237 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Inhibitor REF00000619 DG00251 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Binder REF00000619 DG00290 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Binder REF00002898 DG00303 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Inhibitor REF00001044 DG00313 Bacterial 50S ribosomal RNA (Bact 50S rRNA) . Binder REF00000619 DG00674 Bacterial 50S ribosomal RNA (Bact 50S rRNA) NOUNIPROTAC Modulator REF00003790 DG01168 Bacterial 50S ribosomal RNA (Bact 50S rRNA) NOUNIPROTAC Modulator REF00003421 DG01206 Bacterial 50S ribosomal RNA (Bact 50S rRNA) NOUNIPROTAC Modulator REF00003334 DG01253 Bacterial 50S ribosomal RNA (Bact 50S rRNA) NOUNIPROTAC Modulator REF00003040 DG01515 Bacterial 50S ribosomal RNA (Bact 50S rRNA) NOUNIPROTAC Modulator REF00004360 DG00175 Bacterial 70S ribosomal RNA (Bact 70S rRNA) . Binder REF00001993 DG00335 Bacterial 70S ribosomal RNA (Bact 70S rRNA) . Modulator REF00002472 DG01668 Bacterial 70S ribosomal RNA (Bact 70S rRNA) NOUNIPROTAC Binder REF00004433 DG00183 Bacterial Cell membrane (Bact CM) . Modulator REF00000682 DG01170 Bacterial Cell membrane (Bact CM) NOUNIPROTAC Modulator REF00003405 DG01308 Bacterial Cell membrane (Bact CM) NOUNIPROTAC Modulator REF00003332 DG01494 Bacterial Cell membrane (Bact CM) NOUNIPROTAC Modulator REF00001038 DG00021 Bacterial DD-carboxypeptidase (Bact vanYB) VANY_ENTFA Inhibitor REF00002804 DG00052 Bacterial DD-carboxypeptidase (Bact vanYB) VANY_ENTFA Inhibitor REF00002268 DG00163 Bacterial DD-carboxypeptidase (Bact vanYB) VANY_ENTFA Inhibitor REF00002688 DG00425 Bacterial DD-carboxypeptidase (Bact vanYB) VANY_ENTFA Inhibitor REF00001956 DG00263 Bacterial Deoxyribonucleic acid (Bact DNA) . Modulator REF00000679 DG00445 Bacterial Deoxyribonucleic acid (Bact DNA) . Modulator REF00000663 DG00575 Bacterial Deoxyribonucleic acid (Bact DNA) NOUNIPROTAC Binder REF00003338 DG00647 Bacterial Deoxyribonucleic acid (Bact DNA) NOUNIPROTAC Binder REF00003182 DG00856 Bacterial Deoxyribonucleic acid (Bact DNA) NOUNIPROTAC Binder REF00003439 DG00048 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Inhibitor REF00002688 DG00066 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Binder REF00002037 DG00100 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Binder REF00000942 DG00258 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Inhibitor REF00000608 DG00444 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Binder REF00002729 DG00569 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Inhibitor REF00003337 DG00812 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Inhibitor REF00003161 DG00816 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Inhibitor REF00003178 DG01020 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Inhibitor REF00003520 DG01183 Bacterial Dihydropteroate synthetase (Bact folP) DHPS_ECOLI Inhibitor REF00003137 DG00033 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Modulator REF00000713 DG00047 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Modulator REF00000662 DG00209 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Modulator REF00001425 DG00225 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Modulator REF00001565 DG00240 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Modulator REF00001905 DG00318 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Modulator REF00000713 DG00319 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Inhibitor REF00001130 DG00818 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Inhibitor REF00003126 DG00941 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Inhibitor REF00003425 DG00975 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Inhibitor REF00003424 DG01203 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Inhibitor REF00003136 DG01216 Bacterial DNA gyrase (Bact gyrase) GYRA_STAAU; GYRB_STAAU Inhibitor REF00003442 DG00291 Bacterial DNA gyrase B (Bact gyrB) GYRB_ECOLI Inhibitor REF00002900 DG00319 Bacterial DNA topoisomerase 4A (Bact parC) PARC_ECOLI Inhibitor REF00001130 DG00136 Bacterial Fatty acid synthetase I (Bact inhA) INHA_MYCTU Inhibitor REF00001674 DG00681 Bacterial Fatty acid synthetase I (Bact inhA) INHA_MYCTU Inhibitor REF00003326 DG01064 Bacterial Fatty acid synthetase I (Bact inhA) INHA_MYCTU Inhibitor REF00003085 DG00169 Bacterial Integral membrane LmrP (Bact lmrP) Q9CDQ3_LACLA Modulator REF00000705 DG00668 Bacterial Isoleucyl-tRNA synthetase (Bact ileS) SYI_ECOLI Modulator REF00003142 DG00016 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00001956 DG00035 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000682 DG00037 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00002688 DG00062 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00002069 DG00067 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00002867 DG00078 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000882 DG00080 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00002077 DG00085 Bacterial Penicillin binding protein (Bact PBP) . Modulator REF00001539 DG00121 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00001034 DG00129 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000749 DG00143 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00002804 DG00156 Bacterial Penicillin binding protein (Bact PBP) . Modulator REF00000540 DG00170 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000770 DG00220 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000682 DG00225 Bacterial Penicillin binding protein (Bact PBP) . Inhibitor REF00001565 DG00227 Bacterial Penicillin binding protein (Bact PBP) . Modulator REF00002688 DG00235 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00002826 DG00239 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000993 DG00252 Bacterial Penicillin binding protein (Bact PBP) . Modulator REF00000656 DG00283 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000540 DG00288 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000770 DG00296 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00002801 DG00299 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00002687 DG00308 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000682 DG00311 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00000540 DG00328 Bacterial Penicillin binding protein (Bact PBP) . Modulator REF00002688 DG00419 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00001956 DG00421 Bacterial Penicillin binding protein (Bact PBP) . Binder REF00001956 DG00587 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003611 DG00882 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003429 DG00912 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003164 DG00919 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003422 DG00948 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003152 DG00979 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00002938 DG01051 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003417 DG01055 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00002992 DG01087 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003864 DG01161 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003859 DG01472 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00003880 DG01493 Bacterial Penicillin binding protein (Bact PBP) NOUNIPROTAC . REF00004195 DG00005 Bacterial Penicillin binding protein 1 (Bact pbp) PBPA_ECOLI; PBPB_ECOLI; PBPC_ECOLI Binder REF00000649 DG00139 Bacterial Penicillin binding protein 2 (Bact mrdA) MRDA_ECOLI Modulator REF00000649 DG00193 Bacterial Penicillin binding protein 2 (Bact mrdA) MRDA_ECOLI Binder REF00002688 DG00904 Bacterial Penicillin binding protein 2 (Bact mrdA) MRDA_ECOLI Binder REF00003415 DG00004 Bacterial Penicillin binding protein 3 (Bact mrcA) FTSI_ECOLI Binder REF00000601 DG00005 Bacterial Penicillin binding protein 3 (Bact mrcA) FTSI_ECOLI Binder REF00000649 DG00073 Bacterial Penicillin binding protein 3 (Bact mrcA) FTSI_ECOLI Binder REF00001362 DG00180 Bacterial Penicillin binding protein 3 (Bact mrcA) FTSI_ECOLI Binder REF00000976 DG00207 Bacterial Penicillin binding protein 3 (Bact mrcA) FTSI_ECOLI Binder REF00000540 DG00425 Bacterial Penicillin binding protein 3 (Bact mrcA) FTSI_ECOLI Antagonist REF00001956 DG01186 Bacterial Penicillin binding protein 3 (Bact mrcA) FTSI_ECOLI Antagonist REF00003860 DG00425 Bacterial Penicillin-binding protein 1B (Bact mrcB) PBPB_ECOLI Antagonist REF00001956 DG00265 Bacterial Ribosomal ATPase RbbA (Bact rbbA) RBBA_ECOLI Inhibitor REF00002824 DG01604 Bacterial Ribosomal ATPase RbbA (Bact rbbA) RBBA_ECOLI Inhibitor REF00004359 DG01156 Bacterial RNA polymerase sigma factor SigA (Bact sigA) SIGA_STAA8 Modulator REF00003404 DG00076 Bacterial RNA polymerase switch region (Bact RNAP-SR) . Modulator REF00001245 DG00186 Bacterial RNA polymerase switch region (Bact RNAP-SR) . Inhibitor REF00000662 DG01044 Bacterial UDP-N-acetylglucosamine carboxyvinyltransferase (Bact murA) MURA_ECOLI Inhibitor REF00003366 DG01263 BDNF/NT-3 growth factors receptor (TrkB) NTRK2_HUMAN Modulator REF00003564 DG01439 B-lymphocyte surface antigen B4 (CD19) CD19_HUMAN CAR-T-Cell-Therapy(Dual specific) REF00003239 DG00541 Brentuximab vedotin TNR8_HUMAN Modulator REF00002932 DG00289 Bromodomain-containing protein 2 (BRD2) BRD2_HUMAN Inhibitor REF00001634 DG01596 Bromodomain-containing protein 2 (BRD2) BRD2_HUMAN Inhibitor REF00004241 DG00289 Bromodomain-containing protein 3 (BRD3) BRD3_HUMAN Inhibitor REF00001634 DG01596 Bromodomain-containing protein 3 (BRD3) BRD3_HUMAN Inhibitor REF00004241 DG00289 Bromodomain-containing protein 4 (BRD4) BRD4_HUMAN Inhibitor REF00001634 DG01596 Bromodomain-containing protein 4 (BRD4) BRD4_HUMAN Inhibitor REF00004241 DG01181 Calcineurin (PPP3CA) PP2BA_HUMAN Inhibitor REF00003826 DG01497 Calcineurin (PPP3CA) PP2BA_HUMAN Inhibitor REF00004079 DG01368 Calcitonin gene-related peptide (CALC) NOUNIPROTAC Modulator REF00002965 DG01274 Calcitonin gene-related peptide receptor (CGRPR) CALRL_HUMAN Inhibitor REF00003758 DG01369 Calcitonin gene-related peptide receptor (CGRPR) CALRL_HUMAN Inhibitor REF00003758 DG01376 Calcitonin gene-related peptide receptor (CGRPR) CALRL_HUMAN Inhibitor REF00003758 DG01378 Calcitonin gene-related peptide receptor (CGRPR) CALRL_HUMAN Inhibitor REF00003758 DG00782 Calcium channel unspecific (CaC) NOUNIPROTAC Modulator REF00003047 DG00784 Calcium channel unspecific (CaC) NOUNIPROTAC Modulator REF00003170 DG00098 Calmodulin (CALM) CALM1_HUMAN; CALM2_HUMAN; CALM3_HUMAN Modulator REF00001416 DG00830 Calmodulin (CALM) CALM1_HUMAN; CALM2_HUMAN; CALM3_HUMAN Inhibitor REF00002948 DG01238 cAMP-dependent chloride channel (CFTR) CFTR_HUMAN Activator REF00003254 DG01531 cAMP-dependent chloride channel (CFTR) CFTR_HUMAN Activator REF00004475 DG00084 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Inhibitor REF00001864 DG00131 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Modulator REF00000665 DG00147 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Inhibitor REF00000632 DG00222 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Modulator REF00001657 DG00278 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Modulator REF00000680 DG00914 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Inhibitor REF00003426 DG01054 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Inhibitor REF00003288 DG01081 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Inhibitor REF00003395 DG01137 Candida Cytochrome P450 51 (Candi ERG11) CP51_CANAL Inhibitor REF00003041 DG00013 Candida Squalene epoxidase (Candi ERG1) ERG1_CANAL Modulator REF00002872 DG00003 Candida Thymidylate synthase (Candi TMP1) TYSY_CANAL Inhibitor REF00001109 DG00018 Candida Thymidylate synthase (Candi TMP1) TYSY_CANAL Inhibitor REF00000874 DG00069 Candida Thymidylate synthase (Candi TMP1) TYSY_CANAL Inhibitor REF00000984 DG00225 Candida Thymidylate synthase (Candi TMP1) TYSY_CANAL Inhibitor REF00001977 DG00264 Candida Thymidylate synthase (Candi TMP1) TYSY_CANAL Inhibitor REF00000666 DG00304 Candida Thymidylate synthase (Candi TMP1) TYSY_CANAL Inhibitor REF00001479 DG00849 Candida Thymidylate synthase (Candi TMP1) TYSY_CANAL Inhibitor REF00002957 DG01464 Candida Thymidylate synthase (Candi TMP1) TYSY_CANAL Inhibitor REF00003898 DG01119 Cannabinoid receptor 1 (CB1) CNR1_HUMAN Agonist REF00003631 DG01119 Cannabinoid receptor 2 (CB2) CNR2_HUMAN Activator REF00003631 DG00103 Carbonic anhydrase (CA) . Inhibitor REF00002220 DG00103 Carbonic anhydrase I (CA-I) CAH1_HUMAN Inhibitor REF00002220 DG00735 Carbonic anhydrase I (CA-I) CAH1_HUMAN Inhibitor REF00003553 DG00103 Carbonic anhydrase II (CA-II) CAH2_HUMAN Inhibitor REF00002220 DG00735 Carbonic anhydrase II (CA-II) CAH2_HUMAN Inhibitor REF00003553 DG01117 Carbonic anhydrase II (CA-II) CAH2_HUMAN Inhibitor REF00003819 DG00103 Carbonic anhydrase IV (CA-IV) CAH4_HUMAN Inhibitor REF00002220 DG00952 Carbonic anhydrase IV (CA-IV) CAH4_HUMAN Inhibitor REF00003743 DG00103 Carbonic anhydrase IX (CA-IX) CAH9_HUMAN Inhibitor REF00002220 DG00103 Carbonic anhydrase VI (CA-VI) CAH6_HUMAN Inhibitor REF00002220 DG00103 Carbonic anhydrase XII (CA-XII) CAH12_HUMAN Inhibitor REF00002220 DG00103 Carbonic anhydrase XIV (CA-XIV) CAH14_HUMAN Inhibitor REF00002220 DG00006 Casein kinase II alpha (CSNK2A1) CSK21_HUMAN Inhibitor REF00002102 DG01092 Catechol-O-methyl-transferase (COMT) COMT_HUMAN Inhibitor REF00003631 DG00266 Cationic trypsinogen (PRSS1) TRY1_HUMAN Inhibitor REF00002673 DG01401 C-C chemokine receptor type 4 (CCR4) CCR4_HUMAN Modulator REF00003514 DG01080 C-C chemokine receptor type 5 (CCR5) CCR5_HUMAN Inhibitor REF00003238 DG01080 CCR5 messenger RNA (CCR5 mRNA) CCR5_HUMAN Antagonist REF00003238 DG00326 Cellular tumor antigen p53 (TP53) P53_HUMAN Inhibitor REF00001212 DG00982 Coagulation factor IIa (F2) THRB_HUMAN Inhibitor REF00003500 DG01450 Complement factor H (CFH) CFAH_HUMAN Modulator REF00003667 DG01176 Corticosteroid-binding globulin (SERPINA6) CBG_HUMAN Modulator REF00003438 DG00248 COVID-19 papain-like proteinase (PL-PRO) R1AB_SARS2 (819-2763) Inhibitor REF00001696 DG00644 COVID-19 RNA-directed RNA polymerase (RdRp) R1AB_SARS2 (4393-5324) Inhibitor REF00003436 DG00126 C-X-C chemokine receptor type 2 (CXCR2) CXCR2_HUMAN Modulator REF00000913 DG01477 Cyclin-dependent kinase 2 (CDK2) CDK2_HUMAN Inhibitor REF00004478 DG01264 Cyclin-dependent kinase 4 (CDK4) CDK4_HUMAN Inhibitor REF00002971 DG01265 Cyclin-dependent kinase 4 (CDK4) CDK4_HUMAN Inhibitor REF00003467 DG01266 Cyclin-dependent kinase 4 (CDK4) CDK4_HUMAN Inhibitor REF00002971 DG01291 Cyclin-dependent kinase 4 (CDK4) CDK4_HUMAN Inhibitor REF00003627 DG01576 Cyclin-dependent kinase 4 (CDK4) CDK4_HUMAN Inhibitor REF00004535 DG01617 Cyclin-dependent kinase 4 (CDK4) CDK4_HUMAN Inhibitor REF00001478 DG00006 Cyclin-dependent kinase 6 (CDK6) CDK6_HUMAN Inhibitor REF00002102 DG01264 Cyclin-dependent kinase 6 (CDK6) CDK6_HUMAN Inhibitor REF00002971 DG01265 Cyclin-dependent kinase 6 (CDK6) CDK6_HUMAN Inhibitor REF00003467 DG01266 Cyclin-dependent kinase 6 (CDK6) CDK6_HUMAN Inhibitor REF00002971 DG01291 Cyclin-dependent kinase 6 (CDK6) CDK6_HUMAN Inhibitor REF00003627 DG01576 Cyclin-dependent kinase 6 (CDK6) CDK6_HUMAN Inhibitor REF00004535 DG01617 Cyclin-dependent kinase 6 (CDK6) CDK6_HUMAN Inhibitor REF00001478 DG00865 Cysteine protease (CYP) NOUNIPROTAC Inhibitor REF00003181 DG00006 Cytochrome P450 1B1 (CYP1B1) CP1B1_HUMAN Inhibitor REF00002102 DG00985 Cytoplasmic thioredoxin reductase (TXNRD1) TRXR1_HUMAN Inhibitor REF00003738 DG01388 Cytotoxic T-lymphocyte protein 4 (CTLA-4) CTLA4_HUMAN . REF00003560 DG01385 Dabigatran (Dabi) NOUNIPROTAC Binder REF00003383 DG00142 Dihydrofolate reductase (DHFR) DYR_HUMAN Modulator REF00000904 DG00102 Dihydroorotate dehydrogenase (DHODH) PYRD_HUMAN Modulator REF00002786 DG00069 Dihydrothymine dehydrogenase (DPYD) DPYD_HUMAN Inhibitor REF00000984 DG01464 Dihydrothymine dehydrogenase (DPYD) DPYD_HUMAN Inhibitor REF00003898 DG00103 DNA [cytosine-5]-methyltransferase (DNMT) . Inhibitor REF00002220 DG00860 DNA [cytosine-5]-methyltransferase (DNMT) NOUNIPROTAC Inhibitor REF00003303 DG00103 DNA [cytosine-5]-methyltransferase 3B (DNMT3B) DNM3B_HUMAN Inhibitor REF00002220 DG00023 DNA replication (DNA repli) . Modulator REF00002756 DG00032 DNA topoisomerase I (TOP1) TOP1_HUMAN Modulator REF00002496 DG00052 DNA topoisomerase I (TOP1) TOP1_HUMAN Inhibitor REF00002268 DG00088 DNA topoisomerase I (TOP1) TOP1_HUMAN Modulator REF00001950 DG00090 DNA topoisomerase I (TOP1) TOP1_HUMAN Inhibitor REF00002428 DG00138 DNA topoisomerase I (TOP1) TOP1_HUMAN Modulator REF00001635 DG00281 DNA topoisomerase I (TOP1) TOP1_HUMAN Modulator REF00001997 DG01831 DNA topoisomerase I (TOP1) TOP1_HUMAN Inhibitor REF00004457 DG01850 DNA topoisomerase I (TOP1) TOP1_HUMAN Inhibitor REF00004554 DG00015 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00001463 DG00059 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Inhibitor REF00002876 DG00092 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Inhibitor REF00001908 DG00109 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00002781 DG00148 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00002642 DG00154 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00002780 DG00238 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Inhibitor REF00000839 DG00254 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00001927 DG00257 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Inhibitor REF00001130 DG00413 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Inhibitor REF00000690 DG00702 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00003001 DG00739 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00003858 DG00863 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00003753 DG01025 DNA topoisomerase II (TOP2) TOP2A_HUMAN; TOP2B_HUMAN Modulator REF00003419 DG00064 DNA-directed RNA polymerase (RNAP) . Modulator REF00000580 DG00190 DNA-directed RNA polymerase (RNAP) . Binder REF00000580 DG00025 Dopamine D2 receptor (D2R) DRD2_HUMAN Antagonist REF00000724 DG00162 Dopamine D2 receptor (D2R) DRD2_HUMAN Antagonist REF00000724 DG00580 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003071 DG00731 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003269 DG00795 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003779 DG00800 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003779 DG00823 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003388 DG00824 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003008 DG00868 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003643 DG00922 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003162 DG00994 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003784 DG01311 Dopamine D2 receptor (D2R) DRD2_HUMAN Inhibitor REF00003067 DG00994 Dopamine D3 receptor (D3R) DRD3_HUMAN Antagonist REF00003784 DG00312 Dopamine D4 receptor (D4R) DRD4_HUMAN Modulator REF00001786 DG01562 Dopamine transporter (DAT) SC6A3_HUMAN Inhibitor REF00003900 DG00402 Dual specificity protein phosphatase 1 (DUSP1) DUS1_HUMAN Inhibitor REF00000712 DG00125 Duffy antigen chemokine receptor (ACKR1) ACKR1_HUMAN Modulator REF00002814 DG00211 Duffy antigen chemokine receptor (ACKR1) ACKR1_HUMAN Modulator REF00002815 DG01500 Duffy antigen chemokine receptor (ACKR1) ACKR1_HUMAN Modulator REF00000491 DG01546 E2 ubiquitin-conjugating enzyme T (UBE2T) UBE2T_HUMAN Inhibitor REF00004546 DG01593 EGFR messenger RNA (EGFR mRNA) EGFR_HUMAN Inhibitor REF00004341 DG00842 Elegans Endoprotease bli-4 (Elegans bli-4) BLI4_CAEEL Inhibitor REF00003742 DG01612 Enhancer of zeste homolog 2 (EZH2) EZH2_HUMAN Inhibitor REF00004368 DG01885 Enhancer of zeste homolog 2 (EZH2) EZH2_HUMAN Inhibitor REF00003865 DG00029 Enzyme unspecific (Enz) . Modulator REF00001620 DG00082 Ephrin type-B receptor 4 (EPHB4) EPHB4_HUMAN Modulator REF00001082 DG00120 Epidermal growth factor (EGF) EGF_HUMAN Modulator REF00001187 DG00074 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00002772 DG00101 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00002616 DG00115 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00002460 DG00120 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Modulator REF00001187 DG00137 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00002743 DG00216 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Modulator REF00001900 DG00229 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00001607 DG00244 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00001374 DG00282 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00002738 DG00309 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00001435 DG00316 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00001435 DG00330 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Antagonist REF00002616 DG00340 Epidermal growth factor receptor (EGFR) EGFR_HUMAN . REF00002723 DG00341 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Suppressor REF00001943 DG00619 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Antagonist REF00003376 DG01214 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Antagonist REF00003379 DG01507 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Antagonist REF00004139 DG01539 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Modulator REF00004038 DG01572 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Inhibitor REF00004520 DG01631 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Antagonist REF00004384 DG01663 Epidermal growth factor receptor (EGFR) EGFR_HUMAN Modulator REF00004397 DG00244 ERBB2 messenger RNA (HER2 mRNA) ERBB2_HUMAN Inhibitor REF00001374 DG00074 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN Inhibitor REF00002772 DG00115 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN Inhibitor REF00002460 DG00244 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN Inhibitor REF00001374 DG00309 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN Inhibitor REF00001435 DG00342 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN Inhibitor REF00002067 DG00346 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN . REF00002779 DG01214 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN CAR-T-Cell-Therapy REF00003379 DG01507 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN CAR-T-Cell-Therapy REF00004139 DG01516 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN Inhibitor REF00003969 DG01517 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN CAR-T-Cell-Therapy REF00004294 DG01594 Erbb2 tyrosine kinase receptor (HER2) ERBB2_HUMAN CAR-T-Cell-Therapy REF00004350 DG01901 Erbb3 tyrosine kinase receptor (Erbb-3) ERBB3_HUMAN Modulator REF00004569 DG00309 Erbb4 tyrosine kinase receptor (Erbb-4) ERBB4_HUMAN Inhibitor REF00001435 DG01214 Erbb4 tyrosine kinase receptor (Erbb-4) ERBB4_HUMAN Inhibitor REF00003379 DG00626 ERK activator kinase (MEK) NOUNIPROTAC Inhibitor REF00003718 DG01506 ERK activator kinase 1 (MEK1) MP2K1_HUMAN Inhibitor REF00004364 DG01506 ERK activator kinase 2 (MEK2) MP2K2_HUMAN Inhibitor REF00004364 DG01423 Erythropoietin Receptor (EPOR) EPOR_HUMAN Modulator REF00003342 DG00006 Estradiol 17 beta-dehydrogenase 1 (17-beta-HSD1) DHB1_HUMAN Inhibitor REF00002102 DG00095 Estrogen receptor (ESR) ESR1_HUMAN Antagonist REF00002745 DG00204 Estrogen receptor (ESR) ESR1_HUMAN Antagonist REF00002614 DG00314 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00002709 DG00438 Estrogen receptor (ESR) ESR1_HUMAN Modulator REF00001681 DG00805 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00003715 DG00850 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00003714 DG00895 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00002953 DG01014 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00003573 DG01021 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00003550 DG01046 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00003538 DG01370 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00003677 DG01483 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00004488 DG01785 Estrogen receptor (ESR) ESR1_HUMAN Binder REF00004019 DG00212 Estrogen receptor beta (ESR2) ESR2_HUMAN Modulator REF00001258 DG01014 Estrogen receptor beta (ESR2) ESR2_HUMAN Agonist REF00003573 DG01370 Estrogen receptor beta (ESR2) ESR2_HUMAN Agonist REF00003677 DG00115 Eukaryotic elongation factor 2 kinase (eEF-2K) EF2K_HUMAN Inhibitor REF00002460 DG01010 Extracellular calcium-sensing receptor (CASR) CASR_HUMAN Antagonist REF00003854 DG00627 Extracellular signal-regulated kinase 2 (ERK2) MK01_HUMAN Inhibitor REF00003718 DG01543 Extracellular signal-regulated kinase 2 (ERK2) MK01_HUMAN Inhibitor REF00003978 DG01165 Farnesoid X-activated receptor (FXR) NR1H4_HUMAN Agonist REF00003476 DG00140 Fatty acid amide hydrolase (FAAH) . Inhibitor REF00001692 DG00051 Fatty acid synthase (FASN) FAS_HUMAN Inhibitor REF00002872 DG00581 Fibroblast growth factor (FGF) NOUNIPROTAC Inhibitor REF00003469 DG01625 Fibroblast growth factor (FGF) NOUNIPROTAC Inhibitor REF00004439 DG01883 Fibroblast growth factor (FGF) NOUNIPROTAC Inhibitor REF00004564 DG00550 Fibroblast growth factor receptor (FGFR) NOUNIPROTAC Antagonist REF00003232 DG00581 Fibroblast growth factor receptor (FGFR) NOUNIPROTAC Antagonist REF00003469 DG01595 Fibroblast growth factor receptor (FGFR) NOUNIPROTAC Antagonist REF00004528 DG01597 Fibroblast growth factor receptor (FGFR) NOUNIPROTAC Antagonist REF00003873 DG01613 Fibroblast growth factor receptor (FGFR) NOUNIPROTAC Antagonist REF00004503 DG01625 Fibroblast growth factor receptor (FGFR) NOUNIPROTAC Antagonist REF00004439 DG01653 Fibroblast growth factor receptor (FGFR) NOUNIPROTAC Antagonist REF00004332 DG00128 Fibroblast growth factor receptor 1 (FGFR1) FGFR1_HUMAN Modulator REF00001742 DG00550 Fibroblast growth factor receptor 1 (FGFR1) FGFR1_HUMAN Inhibitor REF00003232 DG01304 Fibroblast growth factor receptor 1 (FGFR1) FGFR1_HUMAN Inhibitor REF00003471 DG01595 Fibroblast growth factor receptor 1 (FGFR1) FGFR1_HUMAN Inhibitor REF00004528 DG01597 Fibroblast growth factor receptor 1 (FGFR1) FGFR1_HUMAN Inhibitor REF00003873 DG01613 Fibroblast growth factor receptor 1 (FGFR1) FGFR1_HUMAN Inhibitor REF00004503 DG01639 Fibroblast growth factor receptor 1 (FGFR1) FGFR1_HUMAN Inhibitor REF00004297 DG01304 Fibroblast growth factor receptor 2 (FGFR2) FGFR2_HUMAN Binder REF00003471 DG01509 Fibroblast growth factor receptor 2 (FGFR2) FGFR2_HUMAN Inhibitor REF00004088 DG01584 Fibroblast growth factor receptor 2 (FGFR2) FGFR2_HUMAN Modulator REF00003999 DG01585 Fibroblast growth factor receptor 2 (FGFR2) FGFR2_HUMAN Binder REF00004094 DG01613 Fibroblast growth factor receptor 2 (FGFR2) FGFR2_HUMAN Binder REF00004503 DG01639 Fibroblast growth factor receptor 2 (FGFR2) FGFR2_HUMAN Binder REF00004297 DG00331 Fibroblast growth factor receptor 3 (FGFR3) FGFR3_HUMAN Inhibitor REF00002205 DG00547 Fibroblast growth factor receptor 3 (FGFR3) FGFR3_HUMAN Inhibitor REF00003232 DG01304 Fibroblast growth factor receptor 3 (FGFR3) FGFR3_HUMAN Inhibitor REF00003471 DG01613 Fibroblast growth factor receptor 3 (FGFR3) FGFR3_HUMAN Inhibitor REF00004503 DG01639 Fibroblast growth factor receptor 3 (FGFR3) FGFR3_HUMAN Inhibitor REF00004297 DG01857 Fibroblast growth factor receptor 3 (FGFR3) FGFR3_HUMAN Inhibitor REF00003956 DG00024 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Binder REF00001267 DG00096 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Inhibitor REF00001061 DG00128 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Inhibitor REF00001742 DG00192 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Modulator REF00002156 DG00429 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Modulator REF00002166 DG00553 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Inhibitor REF00003537 DG01190 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Inhibitor REF00003262 DG01267 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Inhibitor REF00003076 DG01638 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Inhibitor REF00003918 DG01640 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Inhibitor REF00004375 DG01644 Fms-like tyrosine kinase 3 (FLT-3) FLT3_HUMAN Inhibitor REF00004553 DG00012 "Fungal 1,3-beta-glucan synthase (Fung GSC2)" FKS2_YEAST Modulator REF00000701 DG00036 "Fungal 1,3-beta-glucan synthase (Fung GSC2)" FKS2_YEAST Inhibitor REF00002342 DG00079 "Fungal 1,3-beta-glucan synthase (Fung GSC2)" FKS2_YEAST Modulator REF00002342 DG00185 "Fungal 1,3-beta-glucan synthase (Fung GSC2)" FKS2_YEAST Modulator REF00002342 DG01478 "Fungal 1,3-beta-glucan synthase (Fung GSC2)" FKS2_YEAST Modulator REF00004522 DG00572 Fungal Cell membrane ergosterol (Fung CME) NOUNIPROTAC Modulator REF00003217 DG01031 Fungal Microtubule (Fung MicroTU) NOUNIPROTAC Inducer REF00003159 DG00007 Fusion protein Bcr-Abl (Bcr-Abl) BCR_HUMAN-ABL1_HUMAN Modulator REF00002561 DG00144 Fusion protein Bcr-Abl (Bcr-Abl) BCR_HUMAN-ABL1_HUMAN Inhibitor REF00002747 DG00174 Fusion protein Bcr-Abl (Bcr-Abl) BCR_HUMAN-ABL1_HUMAN Inhibitor REF00002561 DG00174 Fyn tyrosine protein kinase (FYN) FYN_HUMAN Inhibitor REF00002561 DG00839 GABA transaminase (ABAT) GABT_HUMAN Inhibitor REF00003440 DG00649 GABA(A) receptor alpha-1 (GABRA1) GBRA1_HUMAN Inhibitor REF00003027 DG00898 GABA(A) receptor alpha-1 (GABRA1) GBRA1_HUMAN Inhibitor REF00003689 DG01771 GABA(A) receptor alpha-1 (GABRA1) GBRA1_HUMAN Inhibitor REF00004192 DG01067 GABA(A) receptor gamma-3 (GABRG3) GBRG3_HUMAN Modulator REF00003656 DG00595 Gamma-aminobutyric acid receptor (GAR) NOUNIPROTAC Inhibitor REF00003593 DG01185 Gastric H(+)/K(+) ATPase (Proton pump) ATP4A_HUMAN; ATP4B_HUMAN Modulator REF00002959 DG00804 Gastric H(+)/K(+) ATPase alpha (ATP4A) ATP4A_HUMAN Modulator REF00003030 DG01840 Gastrin/cholecystokinin type B receptor (CCKBR) GASR_HUMAN Inhibitor REF00003897 DG00540 Gemtuzumab ozogamicin CD33_HUMAN . REF00002930 DG00789 Geranyltranstransferase (FDPS) FPPS_HUMAN Inhibitor REF00003848 DG01262 Glucagon-like peptide 1 receptor (GLP1R) GLP1R_HUMAN Agonist REF00003361 DG00164 Glucocorticoid receptor (NR3C1) GCR_HUMAN Modulator REF00001246 DG00199 Glucocorticoid receptor (NR3C1) GCR_HUMAN Agonist REF00002633 DG00200 Glucocorticoid receptor (NR3C1) GCR_HUMAN Agonist REF00002633 DG00610 Glucocorticoid receptor (NR3C1) GCR_HUMAN Inhibitor REF00003094 DG00611 Glucocorticoid receptor (NR3C1) GCR_HUMAN Inhibitor REF00003094 DG00612 Glucocorticoid receptor (NR3C1) GCR_HUMAN Inhibitor REF00003094 DG00924 Glucocorticoid receptor (NR3C1) GCR_HUMAN Inhibitor REF00003693 DG01015 Glucocorticoid receptor (NR3C1) GCR_HUMAN Inhibitor REF00003735 DG01033 Glucocorticoid receptor (NR3C1) GCR_HUMAN Inhibitor REF00003797 DG01794 Glucocorticoid receptor (NR3C1) GCR_HUMAN Inhibitor REF00004452 DG00641 Glutamate receptor ionotropic kainate 1 (GRIK1) GRIK1_HUMAN Antagonist REF00003593 DG00847 Glutamate receptor ionotropic NMDA 1 (NMDAR1) NMDZ1_HUMAN Agonist REF00003336 DG01816 Glutathione S-transferase omega-1 (GSTO-1) GSTO1_HUMAN Inhibitor REF00004017 DG00657 Glutathione-dependent PGD synthase (HPGDS) HPGDS_HUMAN Inhibitor REF00003006 DG00638 Glycogen synthase kinase-3 alpha (GSK-3A) GSK3A_HUMAN Inhibitor REF00003593 DG01321 Glycoprotein IIb/IIIa receptor (GPIIb/IIIa) ITA2B_HUMAN; ITB3_HUMAN Binder REF00003671 DG01773 Glycoprotein IIb/IIIa receptor (GPIIb/IIIa) ITA2B_HUMAN; ITB3_HUMAN Binder REF00004159 DG01429 GMCSFR-alpha (CSF2RA) CSF2R_HUMAN Stimulator REF00003658 DG01234 Gonadotropin-releasing hormone receptor (GNRHR) GNRHR_HUMAN Modulator REF00003811 DG01819 Gonadotropin-releasing hormone receptor (GNRHR) GNRHR_HUMAN Modulator REF00004534 DG01232 Growth hormone-releasing hormone receptor (GHRHR) GHRHR_HUMAN Agonist REF00003622 DG01236 Growth hormone-releasing hormone receptor (GHRHR) GHRHR_HUMAN Agonist REF00003567 DG00414 Guanylate cyclase (GC) . Inhibitor REF00000712 DG01495 Heat shock protein 90 alpha (HSP90A) HS90A_HUMAN Inhibitor REF00003921 DG01669 Heat shock protein 90 alpha (HSP90A) HS90A_HUMAN Inhibitor REF00004366 DG00278 Hedgehog signaling pathway (HS pathway) . Inhibitor REF00000680 DG01547 Hedgehog signaling pathway (HS pathway) NOUNIPROTAC Inhibitor REF00004355 DG00157 Hepatitis B virus Polymerase (HBV P) Q67889_HBV Inhibitor REF00001139 DG00210 Hepatitis B virus Reverse transcriptase (HBV RT) DPOL_HBVA3 Modulator REF00001139 DG00563 Hepatitis C virus Non-structural 5A (HCV NS5A) POLG_HCV1 Inhibitor REF00002990 DG00564 Hepatitis C virus Non-structural 5A (HCV NS5A) POLG_HCV1 Inhibitor REF00002990 DG00565 Hepatitis C virus Non-structural 5A (HCV NS5A) POLG_HCV1 Inhibitor REF00002990 DG00568 Hepatitis C virus Non-structural 5A (HCV NS5A) POLG_HCV1 Inhibitor REF00002990 DG01551 Hepatitis C virus Non-structural 5A (HCV NS5A) POLG_HCV1 Inhibitor REF00004357 DG01600 Hepatitis C virus Non-structural 5A (HCV NS5A) POLG_HCV1 Inhibitor REF00004556 DG00605 Hepatitis C virus NS3 helicase (HCV NS3) POLG_HCV1 . REF00002990 DG01643 Hepatitis C virus NS3 helicase (HCV NS3) POLG_HCV1 . REF00003933 DG00584 Hepatitis C virus RNA-directed RNA polymerase (HCV NS5B) POLG_HCV1 Modulator REF00002990 DG00585 Hepatitis C virus RNA-directed RNA polymerase (HCV NS5B) POLG_HCV1 Modulator REF00003402 DG00568 Hepatitis C virus Serine protease NS3/4A (HCV NS3/4A) POLG_HCV1 Modulator REF00002990 DG00603 Hepatitis C virus Serine protease NS3/4A (HCV NS3/4A) POLG_HCV1 Modulator REF00002990 DG00604 Hepatitis C virus Serine protease NS3/4A (HCV NS3/4A) POLG_HCV1 Modulator REF00003116 DG00607 Hepatitis C virus Serine protease NS3/4A (HCV NS3/4A) POLG_HCV1 Modulator REF00002990 DG01510 Hepatitis C virus Serine protease NS3/4A (HCV NS3/4A) POLG_HCV1 Modulator REF00003967 DG00008 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00001139 DG00112 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00001662 DG00260 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00001649 DG00588 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00003310 DG00589 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00003310 DG00590 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00003053 DG00591 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00003053 DG00662 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00003354 DG01310 Herpes simplex virus DNA polymerase UL30 (HSV UL30) DPOL_HHV11 Inhibitor REF00003509 DG00050 HGF/Met signaling pathway (HGF/Met pathway) . Inhibitor REF00002690 DG01520 HGF/Met signaling pathway (HGF/Met pathway) NOUNIPROTAC . REF00004563 DG00019 Histamine H1 receptor (H1R) HRH1_HUMAN Antagonist REF00002801 DG00149 Histamine H1 receptor (H1R) HRH1_HUMAN Antagonist REF00000756 DG00727 Histamine H1 receptor (H1R) HRH1_HUMAN Agonist REF00003655 DG00802 Histamine H1 receptor (H1R) HRH1_HUMAN Agonist REF00003762 DG00999 Histamine H1 receptor (H1R) HRH1_HUMAN Agonist REF00003756 DG01066 Histamine H1 receptor (H1R) HRH1_HUMAN Agonist REF00003755 DG01107 Histamine H1 receptor (H1R) HRH1_HUMAN Agonist REF00003547 DG00058 Histamine N-methyltransferase (HNMT) HNMT_HUMAN Inhibitor REF00002814 DG00727 Histamine N-methyltransferase (HNMT) HNMT_HUMAN Inhibitor REF00003655 DG00224 Histone deacetylase (HDAC) . Inhibitor REF00001135 DG00277 Histone deacetylase (HDAC) . Modulator REF00001287 DG00638 Histone deacetylase (HDAC) NOUNIPROTAC Inhibitor REF00003593 DG00176 Histone deacetylase 1 (HDAC1) HDAC1_HUMAN Inhibitor REF00001479 DG01182 Histone deacetylase 1 (HDAC1) HDAC1_HUMAN Inhibitor REF00003466 DG00102 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00002786 DG00203 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00002801 DG00548 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00003016 DG00920 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00003477 DG00937 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00003360 DG01041 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00003530 DG01042 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00003195 DG01197 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00003154 DG01800 HMG-CoA reductase (HMGCR) HMDH_HUMAN Inhibitor REF00003906 DG00002 Human Deoxyribonucleic acid (hDNA) . Modulator REF00002538 DG00020 Human Deoxyribonucleic acid (hDNA) . Binder REF00002321 DG00023 Human Deoxyribonucleic acid (hDNA) . Intercalator REF00002756 DG00081 Human Deoxyribonucleic acid (hDNA) . Breaker REF00001330 DG00153 Human Deoxyribonucleic acid (hDNA) . Modulator REF00002727 DG00159 Human Deoxyribonucleic acid (hDNA) . Modulator REF00002638 DG00273 Human Deoxyribonucleic acid (hDNA) . Modulator REF00002251 DG00294 Human Deoxyribonucleic acid (hDNA) . Modulator REF00002751 DG00297 Human Deoxyribonucleic acid (hDNA) . Binder REF00002542 DG00300 Human Deoxyribonucleic acid (hDNA) . Modulator REF00002773 DG00305 Human Deoxyribonucleic acid (hDNA) . Breaker REF00002491 DG00324 Human Deoxyribonucleic acid (hDNA) . Modulator REF00001753 DG00337 Human Deoxyribonucleic acid (hDNA) . Modulator REF00002681 DG00396 Human Deoxyribonucleic acid (hDNA) . Binder (minor groove binder) REF00000708 DG00434 Human Deoxyribonucleic acid (hDNA) . Modulator REF00002212 DG00752 Human Deoxyribonucleic acid (hDNA) NOUNIPROTAC Binder (minor groove binder) REF00003734 DG00984 Human Deoxyribonucleic acid (hDNA) NOUNIPROTAC Binder (minor groove binder) REF00003714 DG01110 Human Deoxyribonucleic acid (hDNA) NOUNIPROTAC Binder (minor groove binder) REF00003246 DG01256 Human Deoxyribonucleic acid (hDNA) NOUNIPROTAC Binder (minor groove binder) REF00003681 DG01796 Human Deoxyribonucleic acid (hDNA) NOUNIPROTAC Binder (minor groove binder) REF00004172 DG01814 Human Deoxyribonucleic acid (hDNA) NOUNIPROTAC Modulator REF00004205 DG00333 Human immunodeficiency virus Envelope messenger RNA (HIV env mRNA) ENV_HV1H2 . REF00001358 DG00011 Human immunodeficiency virus Integrase (HIV IN) POL_HV1B1 Modulator REF00002775 DG00116 Human immunodeficiency virus Integrase (HIV IN) POL_HV1B1 Inhibitor REF00002782 DG00197 Human immunodeficiency virus Integrase (HIV IN) POL_HV1B1 Modulator REF00002775 DG00246 Human immunodeficiency virus Integrase (HIV IN) POL_HV1B1 Modulator REF00002775 DG00325 Human immunodeficiency virus Integrase (HIV IN) POL_HV1B1 Inhibitor REF00002775 DG00433 Human immunodeficiency virus Integrase (HIV IN) POL_HV1B1 Modulator REF00000712 DG00044 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Modulator REF00001611 DG00091 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Modulator REF00001700 DG00178 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Modulator REF00001358 DG00181 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00001358 DG00279 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00000610 DG00287 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00001700 DG00576 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00003268 DG00577 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00003268 DG00600 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00002990 DG00602 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00002990 DG00606 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00002990 DG01475 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00003940 DG01529 Human immunodeficiency virus Protease (HIV PR) POL_HV1B1 Inhibitor REF00004367 DG00024 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00001267 DG00075 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00001267 DG00089 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Modulator REF00000686 DG00105 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Modulator REF00000790 DG00141 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00001267 DG00166 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00001139 DG00226 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Modulator REF00001267 DG00269 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00001267 DG00315 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00001267 DG00325 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00002775 DG00578 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00003095 DG00888 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00003637 DG00939 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00003412 DG01286 Human immunodeficiency virus Reverse transcriptase (HIV RT) POL_HV1B1 Inhibitor REF00003413 DG01616 HUMAN mammalian target of rapamycin (mTOR) MTOR_HUMAN Inhibitor REF00004194 DG00292 Inactive rhomboid protein 2 (RHBDF2) RHDF2_HUMAN . REF00002044 DG00402 "Indoleamine 2,3-dioxygenase 1 (IDO1)" I23O1_HUMAN Inhibitor REF00000712 DG00851 "Indoleamine 2,3-dioxygenase 1 (IDO1)" I23O1_HUMAN Inhibitor REF00003167 DG01002 Influenza Hemagglutinin (Influ HA) HEMA_I34A1 Inhibitor REF00003525 DG00621 Influenza M2 protein (Influ M) M2_I34A1 Inhibitor REF00003166 DG00622 Influenza M2 protein (Influ M) M2_I34A1 Inhibitor REF00003166 DG00006 Influenza Neuraminidase (Influ NA) NRAM_I33A0 Inhibitor REF00002102 DG00608 Influenza Neuraminidase (Influ NA) NRAM_I33A0 Inhibitor REF00003434 DG01008 Influenza Neuraminidase (Influ NA) NRAM_I33A0 Inhibitor REF00003414 DG01824 Influenza Neuraminidase (Influ NA) NRAM_I33A0 Inhibitor REF00003895 DG00108 Inhibitor of nuclear factor kappa-B kinase beta (IKKB) IKKB_HUMAN Inhibitor REF00002717 DG00217 Inhibitor of nuclear factor kappa-B kinase beta (IKKB) IKKB_HUMAN Inhibitor REF00002595 DG00040 Inosine-5'-monophosphate dehydrogenase (IMPDH) . Intercalator REF00001406 DG00134 Inosine-5'-monophosphate dehydrogenase 1 (IMPDH1) IMDH1_HUMAN Inhibitor REF00001406 DG00194 Inosine-5'-monophosphate dehydrogenase 1 (IMPDH1) IMDH1_HUMAN Inhibitor REF00004633 DG01053 Inosine-5'-monophosphate dehydrogenase 1 (IMPDH1) IMDH1_HUMAN Inhibitor REF00003862 DG00542 Inotuzumab ozogamicin CD22_HUMAN . REF00002933 DG00253 Insulin receptor (INSR) INSR_HUMAN Inhibitor REF00001979 DG01847 Insulin receptor (INSR) INSR_HUMAN Modulator REF00003899 DG00215 Insulin-degrading enzyme (IDE) IDE_HUMAN Inhibitor REF00001181 DG01664 Insulin-like growth factor I receptor (IGF1R) IGF1R_HUMAN Modulator REF00004497 DG01854 Insulin-like growth factor I receptor (IGF1R) IGF1R_HUMAN Antagonist REF00004497 DG01305 Integrin alpha-4/beta-7 (ITGA4/B7) ITA4_HUMAN-ITB7_HUMAN Modulator REF00003445 DG01224 Integrin alpha-L (ITGAL) ITAL_HUMAN Modulator REF00003139 DG01224 Intercellular adhesion molecule ICAM-1 (ICAM1) ICAM1_HUMAN Antagonist REF00003139 DG01848 Interferon-alpha 2 (IFNA2) IFNA2_HUMAN Modulator REF00004405 DG01893 Interferon-alpha 2 (IFNA2) IFNA2_HUMAN Modulator REF00003922 DG01436 Interleukin 3 receptor alpha (IL3RA) IL3RA_HUMAN Agonist REF00003491 DG00198 Interleukin-1 beta (IL1B) IL1B_HUMAN Suppressor REF00002391 DG01027 Interleukin-1 beta (IL1B) IL1B_HUMAN Modulator REF00003340 DG00759 Interleukin-12 beta (IL12B) IL12B_HUMAN Modulator REF00003160 DG01466 Interleukin-12 beta (IL12B) IL12B_HUMAN Modulator REF00003942 DG00322 Interleukin-2 (IL2) IL2_HUMAN Inhibitor REF00002049 DG01350 Interleukin-23 (IL23) IL23A_HUMAN . REF00003300 DG01443 Interleukin-23 (IL23) IL23A_HUMAN . REF00003369 DG01443 Interleukin-37 (IL37) IL37_HUMAN Inhibitor REF00003369 DG00909 Intestinal maltase-glucoamylase (MGAM) MGA_HUMAN Modulator REF00003252 DG00980 Inward rectifier potassium channel Kir1.2 (KCNJ10) KCJ10_HUMAN Blocker REF00003105 DG01642 Isocitrate dehydrogenase (IDH) IDHC_HUMAN; IDHP_HUMAN; IDH3A_HUMAN; IDH3B_HUMAN; IDH3G_HUMAN Inhibitor REF00003872 DG00620 Janus kinase 1 (JAK-1) JAK1_HUMAN Inhibitor REF00003699 DG01550 Janus kinase 1 (JAK-1) JAK1_HUMAN Inhibitor REF00004461 DG00620 Janus kinase 2 (JAK-2) JAK2_HUMAN Inhibitor REF00003699 DG01239 Janus kinase 2 (JAK-2) JAK2_HUMAN Inhibitor REF00002953 DG01534 Janus kinase 2 (JAK-2) JAK2_HUMAN Inhibitor REF00003902 DG01536 Janus kinase 2 (JAK-2) JAK2_HUMAN Inhibitor REF00004115 DG01549 Janus kinase 2 (JAK-2) JAK2_HUMAN Inhibitor REF00003930 DG01550 Janus kinase 2 (JAK-2) JAK2_HUMAN Inhibitor REF00004461 DG01575 Janus kinase 2 (JAK-2) JAK2_HUMAN Modulator REF00004327 DG01579 Janus kinase 2 (JAK-2) JAK2_HUMAN Inhibitor REF00004491 DG01501 Janus kinase 3 (JAK-3) JAK3_HUMAN Modulator REF00004196 DG00266 Kallikrein-related peptidase (KLK) . Inhibitor REF00002673 DG00317 Kinesin-like protein KIF11 (KIF11) KIF11_HUMAN Inhibitor REF00002504 DG00010 Lactoylglutathione lyase (GLO1) LGUL_HUMAN Inhibitor REF00002302 DG00174 LCK tyrosine protein kinase (LCK) LCK_HUMAN Inhibitor REF00002561 DG00338 Leukocyte surface antigen Leu-16 (CD20) CD20_HUMAN . REF00002554 DG01062 Leutinizing-hormone-releasing hormone (GNRH1) GON1_HUMAN Inhibitor REF00003811 DG00543 Loncastuximab tesirine CD19_HUMAN Inhibitor REF00002934 DG00693 Long transient receptor potential channel 8 (TRPM8) TRPM8_HUMAN Antagonist REF00003709 DG01462 Long transient receptor potential channel 8 (TRPM8) TRPM8_HUMAN Antagonist REF00004476 DG00010 L-selectin (SELL) LYAM1_HUMAN Inhibitor REF00002302 DG00553 Macrophage colony-stimulating factor 1 receptor (CSF1R) CSF1R_HUMAN Antagonist REF00003537 DG01582 Mammalian target of rapamycin complex 1 (mTORC1) MTOR_HUMAN-RPTOR_HUMAN-LST8_HUMAN-AKTS1_HUMAN-DPTOR_HUMAN Inhibitor REF00004548 DG00205 MAPK/ERK kinase kinase (MAP3K) . Modulator REF00001055 DG00635 MAPK/ERK kinase kinase (MAP3K) NOUNIPROTAC Inhibitor REF00003149 DG00677 MAPK/ERK kinase kinase (MAP3K) NOUNIPROTAC Inhibitor REF00003464 DG01506 MAPK/ERK kinase kinase (MAP3K) NOUNIPROTAC Inhibitor REF00004364 DG01545 MAPK/ERK kinase kinase (MAP3K) NOUNIPROTAC Inhibitor REF00004236 DG01567 MAPK/ERK kinase kinase (MAP3K) NOUNIPROTAC Inhibitor REF00004182 DG01568 MAPK/ERK kinase kinase (MAP3K) NOUNIPROTAC Inhibitor REF00004162 DG01879 MAPK/ERK kinase kinase (MAP3K) NOUNIPROTAC Modulator REF00004300 DG00876 Matrix metalloproteinase (MMP) NOUNIPROTAC Modulator REF00003501 DG01470 Matrix metalloproteinase (MMP) NOUNIPROTAC Modulator REF00004158 DG00103 Matrix metalloproteinase-13 (MMP-13) MMP13_HUMAN Inhibitor REF00002220 DG00103 Matrix metalloproteinase-9 (MMP-9) MMP9_HUMAN Inhibitor REF00002220 DG00144 Mcl-1 messenger RNA (MCL-1 mRNA) MCL1_HUMAN . REF00002747 DG00326 Mdm2 messenger RNA (MDM2 mRNA) MDM2_HUMAN Inhibitor REF00001212 DG01775 Melatonin receptor type 1A (MTNR1A) MTR1A_HUMAN Antagonist REF00004417 DG00644 MERS-CoV RNA-directed RNA polymerase (RdRp) R1AB_CVEMC (4378-5310) Inhibitor REF00003436 DG00173 Mitochondrial rRNA methyltransferase 2 (MRM2) MRM2_HUMAN Inhibitor REF00000572 DG00414 Monoamine oxidase (MAO) . . REF00000712 DG00777 Monoamine oxidase (MAO) NOUNIPROTAC Inhibitor REF00003096 DG00777 Monoamine oxidase type A (MAO-A) AOFA_HUMAN Inhibitor REF00003096 DG01460 Monoamine oxidase type A (MAO-A) AOFA_HUMAN Inhibitor REF00003282 DG00100 Monoamine oxidase type B (MAO-B) AOFB_HUMAN Inhibitor REF00000942 DG01460 Monoamine oxidase type B (MAO-B) AOFB_HUMAN Inhibitor REF00003282 DG00402 M-phase inducer phosphatase 2 (MPIP2) MPIP2_HUMAN Inhibitor REF00000712 DG00103 Multidrug resistance protein (MDR) . Inhibitor REF00002220 DG00724 Muscarinic acetylcholine receptor M1 (CHRM1) ACM1_HUMAN Agonist REF00003704 DG01779 Muscarinic acetylcholine receptor M1 (CHRM1) ACM1_HUMAN Agonist REF00004266 DG00809 Muscarinic acetylcholine receptor M3 (CHRM3) ACM3_HUMAN Agonist REF00003320 DG00977 Muscarinic acetylcholine receptor M3 (CHRM3) ACM3_HUMAN Agonist REF00003496 DG01035 Muscarinic acetylcholine receptor M3 (CHRM3) ACM3_HUMAN Agonist REF00003153 DG00831 Muscarinic acetylcholine receptor M4 (CHRM4) ACM4_HUMAN Inhibitor REF00003169 DG00801 Muscarinic acetylcholine receptor M5 (CHRM5) ACM5_HUMAN Modulator REF00003861 DG00678 Mycobacterium Arabinosyltransferase C (MycB embC) EMBC_MYCTU Inhibitor REF00003293 DG00847 Mycobacterium Biosynthetic alanine racemase (MycB alr) ALR_MYCSM Inhibitor REF00003336 DG00847 Mycobacterium D-alanine-D-alanine ligase A (MycB ddl) DDL_MYCTU Inhibitor REF00003336 DG01050 Mycobacterium Mycolic acid synthase (MycB cma) CMAS1_MYCTU; CMAS2_MYCTU; CMAS3_MYCTU Inhibitor REF00003331 DG01156 Mycobacterium RNA polymerase (MycB RNAP) RPOA_MYCTU; RPOB_MYCTU; RPOC_MYCTU; RPOZ_MYCTU Inhibitor REF00003404 DG01366 Nectin cell adhesion molecule 4 (NECTIN4) NECT4_HUMAN . REF00003279 DG00933 Neuronal acetylcholine receptor alpha (NACHRA) NOUNIPROTAC Antagonist REF00003348 DG00593 Neuronal acetylcholine receptor alpha-2 (CHRNA2) ACHA2_HUMAN Modulator (allosteric modulator) REF00003744 DG01140 Neuronal acetylcholine receptor alpha-2 (CHRNA2) ACHA2_HUMAN Modulator (allosteric modulator) REF00003433 DG01295 Neutral endopeptidase (MME) NEP_HUMAN CAR-T-Cell-Therapy(Dual specific) REF00003325 DG00768 Nicotinic acetylcholine receptor (nAChR) NOUNIPROTAC Agonist REF00003179 DG00103 Nitric-oxide synthase inducible (NOS2) NOS2_HUMAN Inhibitor REF00002220 DG00847 N-methyl-D-aspartate receptor (NMDAR) NOUNIPROTAC Antagonist REF00003336 DG01782 N-methyl-D-aspartate receptor (NMDAR) NOUNIPROTAC Antagonist REF00004163 DG00767 Norepinephrine transporter (NET) SC6A2_HUMAN Inhibitor REF00002997 DG00855 Norepinephrine transporter (NET) SC6A2_HUMAN Inhibitor REF00003804 DG00946 Norepinephrine transporter (NET) SC6A2_HUMAN Inhibitor REF00003802 DG01778 Norepinephrine transporter (NET) SC6A2_HUMAN Inhibitor REF00004415 DG01846 Norepinephrine transporter (NET) SC6A2_HUMAN Antagonist REF00004336 DG01263 NT-3 growth factor receptor (TrkC) NTRK3_HUMAN Inhibitor REF00003564 DG00039 Nuclear factor NF-kappa-B (NFKB) NFKB1_HUMAN; NFKB2_HUMAN; TF65_HUMAN; RELB_HUMAN; REL_HUMAN Activator REF00002801 DG00217 Nuclear factor NF-kappa-B (NFKB) NFKB1_HUMAN; NFKB2_HUMAN; TF65_HUMAN; RELB_HUMAN; REL_HUMAN Inhibitor REF00002595 DG01460 Nuclear factor NF-kappa-B (NFKB) NFKB1_HUMAN; NFKB2_HUMAN; TF65_HUMAN; RELB_HUMAN; REL_HUMAN Activator REF00003282 DG00573 Onchocerca Glutamate-gated chloride channel (Onchoc GluCl) Q25634_ONCVO Activator REF00003588 DG00132 Opioid receptor (OPR) . Agonist REF00002396 DG00158 Opioid receptor delta (OPRD1) OPRD_HUMAN Binder REF00002396 DG01114 Opioid receptor delta (OPRD1) OPRD_HUMAN Agonist REF00003396 DG01121 Opioid receptor delta (OPRD1) OPRD_HUMAN Agonist REF00003578 DG01143 Opioid receptor delta (OPRD1) OPRD_HUMAN Agonist REF00003632 DG01467 Opioid receptor delta (OPRD1) OPRD_HUMAN Agonist REF00004122 DG01082 Opioid receptor kappa (OPRK1) OPRK_HUMAN Agonist REF00003362 DG00168 Opioid receptor mu (MOP) OPRM_HUMAN Modulator REF00001663 DG01121 Opioid receptor mu (MOP) OPRM_HUMAN Inhibitor REF00003578 DG01825 Opioid receptor mu (MOP) OPRM_HUMAN Inhibitor REF00004416 DG00030 Organic anion transporter M1 (SLCO4C1) SO4C1_HUMAN Modulator REF00001043 DG01126 Oxytocin receptor (OTR) OXYR_HUMAN Antagonist REF00003820 DG01489 Oxytocin receptor (OTR) OXYR_HUMAN Antagonist REF00004539 DG00549 P2Y purinoceptor 12 (P2RY12) P2Y12_HUMAN Antagonist REF00003016 DG01180 P2Y purinoceptor 12 (P2RY12) P2Y12_HUMAN Antagonist REF00003665 DG00737 Peroxisome proliferator-activated receptor alpha (PPARA) PPARA_HUMAN Modulator REF00003165 DG01189 Peroxisome proliferator-activated receptor alpha (PPARA) PPARA_HUMAN Modulator REF00003787 DG01189 Peroxisome proliferator-activated receptor gamma (PPAR-gamma) PPARG_HUMAN Agonist REF00003787 DG01783 Peroxisome proliferator-activated receptor gamma (PPAR-gamma) PPARG_HUMAN Agonist REF00004479 DG01038 Phosphodiesterase 1 (PDE1) NOUNIPROTAC Inhibitor REF00003350 DG00717 Phosphodiesterase 3 (PDE3) NOUNIPROTAC Inhibitor REF00003012 DG00748 Phosphodiesterase 3 (PDE3) NOUNIPROTAC Inhibitor REF00003737 DG00717 Phosphodiesterase 3A (PDE3A) PDE3A_HUMAN Inhibitor REF00003012 DG01314 Phosphodiesterase 3A (PDE3A) PDE3A_HUMAN Inhibitor REF00003714 DG00748 Phosphodiesterase 4 (PDE4) NOUNIPROTAC Inhibitor REF00003737 DG00791 Phosphodiesterase 4D (PDE4D) PDE4D_HUMAN Inhibitor REF00003458 DG01468 Phosphodiesterase 4D (PDE4D) PDE4D_HUMAN Inhibitor REF00004485 DG00659 Phosphodiesterase 5A (PDE5A) PDE5A_HUMAN Inhibitor REF00003590 DG00791 Phosphodiesterase 5A (PDE5A) PDE5A_HUMAN Inhibitor REF00003458 DG01468 Phosphodiesterase 5A (PDE5A) PDE5A_HUMAN Inhibitor REF00004485 DG00661 Phospholipase A2 (PLA2G1B) PA21B_HUMAN Modulator REF00003589 DG01794 Phospholipase A2 (PLA2G1B) PA21B_HUMAN Modulator REF00004452 DG00045 PI3K/AKT/mTOR pathway (PAm pathway) . Inhibitor REF00002046 DG00284 PI3-kinase alpha (PIK3CA) PK3CA_HUMAN Inhibitor REF00001844 DG01270 PI3-kinase alpha (PIK3CA) PK3CA_HUMAN Inhibitor REF00003529 DG01533 PI3-kinase alpha (PIK3CA) PK3CA_HUMAN Inhibitor REF00004523 DG01592 PI3-kinase alpha (PIK3CA) PK3CA_HUMAN Inhibitor REF00004341 DG01671 PI3-kinase alpha (PIK3CA) PK3CA_HUMAN Inhibitor REF00004373 DG01871 PI3-kinase alpha (PIK3CA) PK3CA_HUMAN Inhibitor REF00004016 DG01533 PI3-kinase beta (PIK3CB) PK3CB_HUMAN Inhibitor REF00004523 DG01565 PI3-kinase beta (PIK3CB) PK3CB_HUMAN Modulator REF00004551 DG01566 PI3-kinase beta (PIK3CB) PK3CB_HUMAN Inhibitor REF00004103 DG00648 PI3-kinase delta (PIK3CD) PK3CD_HUMAN Inhibitor REF00003563 DG01270 PI3-kinase delta (PIK3CD) PK3CD_HUMAN Inhibitor REF00003529 DG01271 PI3-kinase delta (PIK3CD) PK3CD_HUMAN Inhibitor REF00003529 DG01533 PI3-kinase delta (PIK3CD) PK3CD_HUMAN Inhibitor REF00004523 DG01587 PI3-kinase delta (PIK3CD) PK3CD_HUMAN Inhibitor REF00004815 DG01671 PI3-kinase delta (PIK3CD) PK3CD_HUMAN Inhibitor REF00004373 DG00280 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Modulator REF00001567 DG00545 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00003377 DG01270 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00003529 DG01271 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00003529 DG01533 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004523 DG01537 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004101 DG01548 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00003930 DG01552 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004294 DG01557 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004037 DG01570 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004392 DG01582 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004548 DG01587 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004815 DG01592 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004341 DG01671 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004373 DG01869 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Modulator REF00003948 DG01876 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004353 DG01877 PI3-kinase gamma (PIK3CG) PK3CG_HUMAN Inhibitor REF00004187 DG00191 Plasmodium 80S ribosome (Malaria 80S) . Binder REF00002814 DG00006 Plasmodium CDK Pfmrk (Malaria Pfmrk) P90584_PLAFA Inhibitor REF00002102 DG00102 Plasmodium Dihydroorotate dehydrogenase (Malaria DHOdehase) PYRD_PLAF7 Inhibitor REF00002786 DG00262 Plasmodium Dihydroorotate dehydrogenase (Malaria DHOdehase) PYRD_PLAF7 Inhibitor REF00002143 DG00402 Plasmodium Dihydroorotate dehydrogenase (Malaria DHOdehase) PYRD_PLAF7 Inhibitor REF00000712 DG00551 Plasmodium Dihydroorotate dehydrogenase (Malaria DHOdehase) PYRD_PLAF7 Inhibitor REF00003094 DG00976 Plasmodium Dihydroorotate dehydrogenase (Malaria DHOdehase) PYRD_PLAF7 Inhibitor REF00003798 DG00687 Plasmodium DOXP reductoisomerase (Malaria DXR) DXR_PLAFX Inhibitor REF00003121 DG00302 Plasmodium Elongation factor 1-alpha 1 (Malaria MEF-1) EF1A_PLAFK Inhibitor REF00000599 DG00001 Plasmodium Enoyl-ACP reductase (Malaria fabI) Q965D5_PLAFA Binder REF00000872 DG00128 Platelet-derived growth factor receptor (PDGFR) . Modulator REF00001742 DG00144 Platelet-derived growth factor receptor (PDGFR) . Inhibitor REF00002747 DG00331 Platelet-derived growth factor receptor (PDGFR) . Inhibitor REF00002205 DG00332 Platelet-derived growth factor receptor (PDGFR) . Inhibitor REF00002310 DG00547 Platelet-derived growth factor receptor (PDGFR) NOUNIPROTAC Inhibitor REF00003232 DG01522 Platelet-derived growth factor receptor (PDGFR) NOUNIPROTAC Inhibitor REF00003966 DG01306 Platelet-derived growth factor receptor alpha (PDGFRA) PGFRA_HUMAN Inhibitor REF00003470 DG01623 Platelet-derived growth factor receptor alpha (PDGFRA) PGFRA_HUMAN Inhibitor REF00003968 DG01624 Platelet-derived growth factor receptor alpha (PDGFRA) PGFRA_HUMAN Inhibitor REF00004392 DG01652 Platelet-derived growth factor receptor alpha (PDGFRA) PGFRA_HUMAN Inhibitor REF00004389 DG00282 Platelet-derived growth factor receptor beta (PDGFRB) PGFRB_HUMAN Modulator REF00002738 DG00219 Pneumocystis carinii Dihydropteroate synthase (PC DHPS) FOL1_PNECA Modulator REF00000679 DG00202 Poly [ADP-ribose] polymerase (PARP) . Modulator REF00001617 DG00334 Poly [ADP-ribose] polymerase (PARP) . Modulator REF00001349 DG01198 Poly [ADP-ribose] polymerase (PARP) NOUNIPROTAC Modulator REF00003245 DG01502 Poly [ADP-ribose] polymerase (PARP) NOUNIPROTAC Modulator REF00004043 DG01538 Poly [ADP-ribose] polymerase (PARP) NOUNIPROTAC Modulator REF00004541 DG01155 Polypeptide deformylase (PDF) DEFM_HUMAN Inhibitor REF00003798 DG01806 PP2A B subunit isoform R5-alpha (PPP2R5A) 2A5A_HUMAN Inhibitor REF00004201 DG00087 Progesterone receptor (PGR) PRGR_HUMAN Agonist REF00002604 DG00867 Progesterone receptor (PGR) PRGR_HUMAN Agonist REF00003539 DG01363 Programmed cell death 1 ligand 1 (PD-L1) PD1L1_HUMAN CAR-T-Cell-Therapy(Dual specific) REF00003472 DG00344 Programmed cell death protein 1 (PD-1) PDCD1_HUMAN . REF00001693 DG01406 Programmed cell death protein 1 (PD-1) PDCD1_HUMAN Inhibitor REF00003698 DG01431 Programmed cell death protein 1 (PD-1) PDCD1_HUMAN Inhibitor REF00003778 DG00010 Prolyl endopeptidase (PREP) PPCE_HUMAN Inhibitor REF00002302 DG01195 Prostacyclin receptor (PTGIR) PI2R_HUMAN Modulator REF00003518 DG00583 Prostaglandin F2-alpha receptor (PTGFR) PF2R_HUMAN Antagonist REF00003314 DG00548 Prostaglandin G/H synthase (COX) PGH1_HUMAN; PGH2_HUMAN Modulator REF00003016 DG00633 Prostaglandin G/H synthase (COX) PGH1_HUMAN; PGH2_HUMAN Modulator REF00002950 DG00762 Prostaglandin G/H synthase (COX) PGH1_HUMAN; PGH2_HUMAN Modulator REF00003630 DG01006 Prostaglandin G/H synthase (COX) PGH1_HUMAN; PGH2_HUMAN Modulator REF00003011 DG01778 Prostaglandin G/H synthase (COX) PGH1_HUMAN; PGH2_HUMAN Modulator REF00004415 DG00103 Prostaglandin G/H synthase 1 (COX-1) PGH1_HUMAN Inhibitor REF00002220 DG00806 Prostaglandin G/H synthase 1 (COX-1) PGH1_HUMAN Inhibitor REF00003029 DG00103 Prostaglandin G/H synthase 2 (COX-2) PGH2_HUMAN Inhibitor REF00002220 DG00613 Prostaglandin G/H synthase 2 (COX-2) PGH2_HUMAN Inhibitor REF00003094 DG00615 Prostaglandin G/H synthase 2 (COX-2) PGH2_HUMAN Inhibitor REF00003614 DG00761 Prostaglandin G/H synthase 2 (COX-2) PGH2_HUMAN Inhibitor REF00003652 DG00995 Prostaglandin G/H synthase 2 (COX-2) PGH2_HUMAN Inhibitor REF00003059 DG00582 Prostaglandin receptor (PTGR) NOUNIPROTAC Modulator REF00003314 DG00266 Proteasome (PS) . Modulator REF00002673 DG01190 Protein kinase C gamma (PRKCG) KPCG_HUMAN Inhibitor REF00003262 DG00255 Proton-coupled folate transporter (SLC46A1) PCFT_HUMAN Modulator REF00002022 DG00267 Proton-coupled folate transporter (SLC46A1) PCFT_HUMAN Modulator REF00002618 DG00050 Proto-oncogene c-Met (MET) MET_HUMAN Modulator REF00002690 DG00213 Proto-oncogene c-Met (MET) MET_HUMAN Inhibitor REF00001925 DG00617 Proto-oncogene c-Met (MET) MET_HUMAN CAR-T-Cell-Therapy(Dual specific) REF00003330 DG01249 Proto-oncogene c-Met (MET) MET_HUMAN CAR-T-Cell-Therapy(Dual specific) REF00003157 DG01498 Proto-oncogene c-Met (MET) MET_HUMAN Inhibitor REF00004487 DG01520 Proto-oncogene c-Met (MET) MET_HUMAN CAR-T-Cell-Therapy(Dual specific) REF00004563 DG01571 Proto-oncogene c-Met (MET) MET_HUMAN Modulator REF00004294 DG01619 Proto-oncogene c-Met (MET) MET_HUMAN CAR-T-Cell-Therapy(Dual specific) REF00004183 DG00192 Proto-oncogene c-Ret (RET) RET_HUMAN Modulator REF00002156 DG00619 Proto-oncogene c-Ret (RET) RET_HUMAN Inhibitor REF00003376 DG01307 Proto-oncogene c-Ret (RET) RET_HUMAN Inhibitor REF00003052 DG01309 Proto-oncogene c-Ret (RET) RET_HUMAN Inhibitor REF00003052 DG01513 Proto-oncogene c-Ret (RET) RET_HUMAN Modulator REF00003968 DG00050 Proto-oncogene c-Ros (ROS1) ROS1_HUMAN Modulator REF00002690 DG01520 Proto-oncogene c-Ros (ROS1) ROS1_HUMAN Inhibitor REF00004563 DG00174 Proto-oncogene c-Src (SRC) SRC_HUMAN Inhibitor REF00002561 DG00214 Proto-oncogene c-Src (SRC) SRC_HUMAN Modulator REF00002406 DG00230 Proto-oncogene c-Src (SRC) SRC_HUMAN Inhibitor REF00001231 DG00010 P-selectin (SELP) LYAM3_HUMAN Inhibitor REF00002302 DG01772 PTPN1 messenger RNA (PTPN1 mRNA) PTN1_HUMAN Inhibitor REF00004075 DG00320 Pyruvate dehydrogenase kinase 1 (PDHK1) PDK1_HUMAN Inhibitor REF00002734 DG01775 Quinone reductase 2 (NQO2) NQO2_HUMAN Inhibitor REF00004417 DG00309 RAC-alpha serine/threonine-protein kinase (AKT1) AKT1_HUMAN Inhibitor REF00001435 DG00652 RAC-alpha serine/threonine-protein kinase (AKT1) AKT1_HUMAN Inhibitor REF00003515 DG01541 RAC-alpha serine/threonine-protein kinase (AKT1) AKT1_HUMAN Inhibitor REF00004130 DG01556 RAC-alpha serine/threonine-protein kinase (AKT1) AKT1_HUMAN Inhibitor REF00004124 DG01577 RAC-alpha serine/threonine-protein kinase (AKT1) AKT1_HUMAN Inhibitor REF00004069 DG01620 RAC-alpha serine/threonine-protein kinase (AKT1) AKT1_HUMAN Inhibitor REF00004532 DG01546 RAC-gamma serine/threonine-protein kinase (AKT3) AKT3_HUMAN Inhibitor REF00004546 DG01555 RAC-gamma serine/threonine-protein kinase (AKT3) AKT3_HUMAN Modulator REF00004276 DG01556 RAC-gamma serine/threonine-protein kinase (AKT3) AKT3_HUMAN Inhibitor REF00004124 DG01583 RAC-gamma serine/threonine-protein kinase (AKT3) AKT3_HUMAN Modulator REF00003901 DG00295 Ras-related protein Rab-9A (RAB9A) RAB9A_HUMAN Inhibitor REF00002113 DG01021 Respiratory syncytial virus protein F (RSV F) FUS_HRSVA Inhibitor REF00003550 DG01412 Respiratory syncytial virus protein F (RSV F) FUS_HRSVA Inhibitor REF00003803 DG00027 Retinoic acid receptor (RAR) . Binder REF00000893 DG00027 Retinoic acid receptor gamma (RARG) RARG_HUMAN Agonist REF00000893 DG00819 Retinoic acid receptor gamma (RARG) RARG_HUMAN Antagonist REF00003031 DG01469 Retinoic acid receptor gamma (RARG) RARG_HUMAN Antagonist REF00004149 DG00049 Ribonucleoside-diphosphate reductase M2 (RRM2) RIR2_HUMAN Modulator REF00002759 DG00746 Ribonucleoside-diphosphate reductase M2 (RRM2) RIR2_HUMAN . REF00003000 DG01873 Ribosomal protein S6 kinase (S6K) NOUNIPROTAC Modulator REF00004191 DG00093 Ribosome A (hRA) . Modulator REF00001260 DG00218 Ribosome A (hRA) . Modulator REF00001291 DG01013 RNA synthesis (hRNA synth) NOUNIPROTAC Modulator REF00003236 DG00402 Rotamase Pin1 (PIN1) PIN1_HUMAN Inhibitor REF00000712 DG01173 Ryanodine receptor (RYR) NOUNIPROTAC Modulator REF00003646 DG00167 Sarcoplasmic/endoplasmic reticulum calcium ATPase (ATP2A) . Inhibitor REF00001754 DG00223 Sarcoplasmic/endoplasmic reticulum calcium ATPase (ATP2A) . Inhibitor REF00002794 DG00232 Sarcoplasmic/endoplasmic reticulum calcium ATPase (ATP2A) . Inhibitor REF00002531 DG00262 Sarcoplasmic/endoplasmic reticulum calcium ATPase (ATP2A) . Inhibitor REF00002143 DG00645 Sarcoplasmic/endoplasmic reticulum calcium ATPase (ATP2A) NOUNIPROTAC Inhibitor REF00003321 DG01835 Sarcoplasmic/endoplasmic reticulum calcium ATPase (ATP2A) NOUNIPROTAC Inhibitor REF00003895 DG00644 SARS-CoV RNA-directed RNA polymerase (RdRp) R1AB_CVHSA (4370-5301) Inhibitor REF00003436 DG00788 Schistosoma Deoxyribonucleic acid (Schist DNA) NOUNIPROTAC Modulator REF00003598 DG00838 Serine/threonine PP1-alpha (PPP1CA) PP1A_HUMAN Inhibitor REF00003058 DG01806 Serine/threonine PP1-alpha (PPP1CA) PP1A_HUMAN Inhibitor REF00004201 DG01590 Serine/threonine-protein kinase ATR (FRP1) ATR_HUMAN Inhibitor REF00004449 DG01591 Serine/threonine-protein kinase ATR (FRP1) ATR_HUMAN Inhibitor REF00003997 DG01611 Serine/threonine-protein kinase ATR (FRP1) ATR_HUMAN Inhibitor REF00004445 DG00072 Serine/threonine-protein kinase B-raf (BRAF) BRAF_HUMAN Inhibitor REF00002757 DG00306 Serine/threonine-protein kinase B-raf (BRAF) BRAF_HUMAN Modulator REF00002323 DG00642 Serine/threonine-protein kinase B-raf (BRAF) BRAF_HUMAN Inhibitor REF00003462 DG01523 Serine/threonine-protein kinase B-raf (BRAF) BRAF_HUMAN Inhibitor REF00004033 DG01588 Serine/threonine-protein kinase B-raf (BRAF) BRAF_HUMAN Inhibitor REF00004330 DG01641 Serine/threonine-protein kinase B-raf (BRAF) BRAF_HUMAN Inhibitor REF00004000 DG00045 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00002046 DG00177 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00001567 DG00195 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00002686 DG00206 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00001567 DG00208 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00001567 DG00280 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Modulator REF00001567 DG00545 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00003377 DG00628 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00003823 DG01496 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00003936 DG01548 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00003930 DG01570 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00004392 DG01573 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Modulator REF00004527 DG01581 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Modulator REF00004362 DG01582 Serine/threonine-protein kinase mTOR (mTOR) MTOR_HUMAN Inhibitor REF00004548 DG01608 Serine/threonine-protein kinase pim-2 (PIM2) PIM2_HUMAN Modulator REF00004817 DG01628 Serine/threonine-protein kinase Raf (RAF) ARAF_HUMAN; BRAF_HUMAN; RAF1_HUMAN Modulator REF00004139 DG00855 Serotonin transporter (SERT) SC6A4_HUMAN Inhibitor REF00003804 DG00953 Serotonin transporter (SERT) SC6A4_HUMAN Inhibitor REF00003258 DG01778 Serotonin transporter (SERT) SC6A4_HUMAN Inhibitor REF00004415 DG00441 Serum albumin (ALB) ALBU_HUMAN Binder REF00000712 DG01834 Sigma intracellular receptor 2 (TMEM97) SGMR2_HUMAN Antagonist REF00004560 DG00123 Signal transducer and activator of transcription 3 (STAT3) STAT3_HUMAN Inhibitor REF00001537 DG01511 Signal transducer and activator of transcription 3 (STAT3) STAT3_HUMAN Inhibitor REF00003943 DG01823 SLC5A2 messenger RNA (SLC5A2 mRNA) SC5A2_HUMAN Inhibitor REF00004211 DG00813 S-mephenytoin 4-hydroxylase (CYP2C9) CP2C9_HUMAN Modulator REF00003069 DG00042 Smoothened homolog (SMO) SMO_HUMAN Modulator REF00001578 DG00660 Smoothened homolog (SMO) SMO_HUMAN Antagonist REF00003390 DG01540 Smoothened homolog (SMO) SMO_HUMAN Antagonist REF00003996 DG00596 Sodium channel unspecific (NaC) NOUNIPROTAC Blocker REF00003399 DG00637 Sodium channel unspecific (NaC) NOUNIPROTAC Blocker REF00003593 DG00077 Sodium pump subunit alpha-1 (ATP1A1) AT1A1_HUMAN Binder REF00002814 DG00956 Sodium pump subunit alpha-1 (ATP1A1) AT1A1_HUMAN Inhibitor REF00003609 DG01245 Sodium/glucose cotransporter 2 (SGLT2) SC5A2_HUMAN Inhibitor REF00003486 DG00030 Sodium/potassium-transporting ATPase (SPT ATPase) AT1A1_HUMAN; AT1A2_HUMAN; AT1A3_HUMAN; AT1B1_HUMAN; AT1B2_HUMAN; AT1B3_HUMAN Inhibitor REF00001043 DG00405 Sodium/potassium-transporting ATPase (SPT ATPase) AT1A1_HUMAN; AT1A2_HUMAN; AT1A3_HUMAN; AT1B1_HUMAN; AT1B2_HUMAN; AT1B3_HUMAN Modulator REF00002418 DG00267 Solute carrier family 19 member 1 (SLC19A1) S19A1_HUMAN Modulator REF00002618 DG00404 Solute carrier family 22 member 8 (SLC22A8) S22A8_HUMAN Blocker REF00002808 DG00165 Solute carrier family 47 member 1 (SLC47A1) S47A1_HUMAN Modulator REF00002447 DG00843 Somatostatin (SST) SMS_HUMAN Binder REF00003676 DG01047 Somatostatin receptor type 2 (SSTR2) SSR2_HUMAN Antagonist REF00002972 DG00989 Sphingosine-1-phosphate receptor 1 (S1PR1) S1PR1_HUMAN Agonist REF00003431 DG00916 Squalene monooxygenase (SQLE) ERG1_HUMAN Inhibitor REF00003407 DG00031 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00002512 DG00057 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00000730 DG00068 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00001005 DG00094 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00000775 DG00117 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00001892 DG00118 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00002355 DG00187 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00002744 DG00201 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00001892 DG00221 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00000672 DG00259 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00000641 DG00301 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00001539 DG00310 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00000654 DG01091 Staphylococcus 30S ribosomal subunit (Stap-coc pbp2) F4NA87_STAAU Binder REF00003196 DG00998 Staphylococcus Beta-lactamase (Stap-coc blaZ) BLAC_STAAU Inhibitor REF00003441 DG01914 Staphylococcus Enoyl ACP reductase (Stap-coc fabI) FABI_STAA8 Inhibitor REF00004341 DG01212 Staphylococcus Leucyl-tRNA synthetase (Stap-coc leuS) SYL_STAAE Inhibitor REF00003410 DG01156 Staphylococcus Plastid RNA polymerase beta (Stap-coc rpoB) RPOB_STAA8 Inhibitor REF00003404 DG00033 Staphylococcus Topoisomerase IV (Stap-coc parC) PARC_STAAS Modulator REF00000713 DG00209 Staphylococcus Topoisomerase IV (Stap-coc parC) PARC_STAAS Modulator REF00001425 DG00225 Staphylococcus Topoisomerase IV (Stap-coc parC) PARC_STAAS Modulator REF00001977 DG00318 Staphylococcus Topoisomerase IV (Stap-coc parC) PARC_STAAS Modulator REF00000713 DG00818 Staphylococcus Topoisomerase IV (Stap-coc parC) PARC_STAAS Inhibitor REF00003126 DG01203 Staphylococcus Topoisomerase IV (Stap-coc parC) PARC_STAAS Inhibitor REF00003136 DG01216 Staphylococcus Topoisomerase IV (Stap-coc parC) PARC_STAAS Inhibitor REF00003442 DG00034 Steroid 17-alpha-monooxygenase (S17AH) CP17A_HUMAN Modulator REF00001776 DG00884 Steroid hormone receptor ERR (ESRR) ERR1_HUMAN; ERR2_HUMAN; ERR3_HUMAN Modulator REF00003037 DG01037 Steroid hormone receptor ERR (ESRR) ERR1_HUMAN; ERR2_HUMAN; ERR3_HUMAN Modulator REF00003863 DG01242 Steroid hormone receptor ERR (ESRR) ERR1_HUMAN; ERR2_HUMAN; ERR3_HUMAN Modulator REF00003674 DG01107 Steryl-sulfatase (STS) STS_HUMAN Inhibitor REF00003547 DG00667 Streptococcus Elongation factor G (Stre-coc fusA) EFG_STRZJ Inhibitor REF00003850 DG00316 Stress-activated protein kinase 2a (p38 alpha) MK14_HUMAN Inhibitor REF00001435 DG00833 Synaptic vesicle amine transporter (SLC18A2) VMAT2_HUMAN Antagonist REF00003263 DG01299 Synaptic vesicle amine transporter (SLC18A2) VMAT2_HUMAN Antagonist REF00003651 DG01300 Synaptic vesicle amine transporter (SLC18A2) VMAT2_HUMAN Antagonist REF00003651 DG01301 Synaptic vesicle amine transporter (SLC18A2) VMAT2_HUMAN Antagonist REF00003651 DG00640 Synaptic vesicle glycoprotein 2A (SV2A) SV2A_HUMAN Binder REF00003593 DG01582 Target of rapamycin complex 2 MAPKAP1 (MTORC2) SIN1_HUMAN Inhibitor REF00004548 DG01333 T-cell-specific surface glycoprotein CD28 (CD28) CD28_HUMAN CAR-T-Cell-Therapy(Dual specific) REF00003805 DG00285 Telomerase reverse transcriptase (TERT) TERT_HUMAN Inhibitor REF00002668 DG00069 TERT messenger RNA (TERT mRNA) TERT_HUMAN . REF00000984 DG00104 TERT messenger RNA (TERT mRNA) TERT_HUMAN Inhibitor REF00002823 DG00109 TERT messenger RNA (TERT mRNA) TERT_HUMAN . REF00002781 DG01464 TERT messenger RNA (TERT mRNA) TERT_HUMAN . REF00003898 DG00069 Thymidylate synthase messenger RNA (TYMS mRNA) TYSY_HUMAN . REF00000984 DG01464 Thymidylate synthase messenger RNA (TYMS mRNA) TYSY_HUMAN . REF00003898 DG00329 Thyroid hormone receptor alpha (THRA) THA_HUMAN Antagonist REF00002705 DG00654 Thyroid peroxidase (TPO) PERT_HUMAN Modulator REF00003497 DG00897 Thyroid peroxidase (TPO) PERT_HUMAN Modulator REF00003447 DG01442 Thyrotropin receptor (TSHR) TSHR_HUMAN Agonist REF00003060 DG01818 Thyrotropin-releasing hormone receptor (TRHR) TRFR_HUMAN Inhibitor REF00004515 DG01320 T-lymphocyte activation antigen CD86 (FUN1) CD86_HUMAN . REF00003131 DG00928 Toll-like receptor 7 (TLR7) TLR7_HUMAN Antagonist REF00003757 DG00929 Toll-like receptor 7 (TLR7) TLR7_HUMAN Antagonist REF00003757 DG00929 Toll-like receptor 8 (TLR8) TLR8_HUMAN Antagonist REF00003757 DG00196 Transformation-sensitive protein p120 (TRPA1) TRPA1_HUMAN Activator REF00002095 DG00693 Transformation-sensitive protein p120 (TRPA1) TRPA1_HUMAN Antagonist REF00003709 DG01462 Transformation-sensitive protein p120 (TRPA1) TRPA1_HUMAN Antagonist REF00004476 DG00656 Transforming growth factor beta 1 (TGFB1) TGFB1_HUMAN Modulator REF00003490 DG00271 Transient receptor potential cation channel V1 (TRPV1) TRPV1_HUMAN Agonist REF00000618 DG00274 Translocator protein (TSPO) TSPO_HUMAN Modulator REF00002541 DG00699 Translocator protein (TSPO) TSPO_HUMAN Binder REF00003043 DG01263 Tropomyosin-related kinase A (TrkA) NTRK1_HUMAN Inhibitor REF00003564 DG00917 Trypanosoma Cruzipain (Trypano CYSP) CYSP_TRYCR Inhibitor REF00003194 DG00065 Tryptase alpha/beta-1 (Tryptase) TRYB1_HUMAN Inhibitor REF00000676 DG00017 Tubulin (TUB) . Inhibitor REF00001733 DG00124 Tubulin (TUB) . Binder REF00001706 DG00161 Tubulin (TUB) . Inhibitor REF00000814 DG00228 Tubulin (TUB) . Inhibitor REF00002724 DG01191 Tubulin (TUB) NOUNIPROTAC Modulator REF00003728 DG01209 Tubulin (TUB) NOUNIPROTAC Modulator REF00003233 DG01474 Tubulin (TUB) NOUNIPROTAC Modulator REF00004036 DG00133 Tubulin beta (TUBB) . Modulator REF00002761 DG00151 Tubulin beta (TUBB) . Modulator REF00002764 DG00646 Tubulin beta (TUBB) NOUNIPROTAC Inhibitor REF00003824 DG00653 Tubulin beta (TUBB) NOUNIPROTAC Inhibitor REF00003673 DG00908 Tubulin beta (TUBB) NOUNIPROTAC Inhibitor REF00003474 DG00286 Tubulin beta-2 chain (TUBB2) TBB2A_HUMAN Inhibitor REF00001619 DG00010 Tumor necrosis factor (TNF) TNFA_HUMAN Inhibitor REF00002302 DG00198 Tumor necrosis factor (TNF) TNFA_HUMAN Suppressor REF00002391 DG00241 Tumor necrosis factor (TNF) TNFA_HUMAN Inhibitor REF00001318 DG00275 Tumor necrosis factor (TNF) TNFA_HUMAN Inhibitor REF00001727 DG01322 Tumor necrosis factor (TNF) TNFA_HUMAN Inhibitor REF00003300 DG01773 Tyrosinase (TYR) TYRO_HUMAN Inhibitor REF00004159 DG00082 Tyrosine-protein kinase (PTK) . Inhibitor REF00001082 DG00192 Tyrosine-protein kinase ABL1 (ABL) ABL1_HUMAN Modulator REF00002156 DG00214 Tyrosine-protein kinase ABL1 (ABL) ABL1_HUMAN Modulator REF00002406 DG00230 Tyrosine-protein kinase ABL1 (ABL) ABL1_HUMAN Inhibitor REF00001598 DG01578 Tyrosine-protein kinase ABL1 (ABL) ABL1_HUMAN Inhibitor REF00003916 DG00130 Tyrosine-protein kinase BTK (ATK) BTK_HUMAN Inhibitor REF00002763 DG00144 Tyrosine-protein kinase Kit (KIT) KIT_HUMAN Inhibitor REF00002747 DG00192 Tyrosine-protein kinase Kit (KIT) KIT_HUMAN Modulator REF00002156 DG00282 Tyrosine-protein kinase Kit (KIT) KIT_HUMAN Modulator REF00002738 DG00332 Tyrosine-protein kinase Kit (KIT) KIT_HUMAN Inhibitor REF00002310 DG00553 Tyrosine-protein kinase Kit (KIT) KIT_HUMAN Inhibitor REF00003537 DG01522 Tyrosine-protein kinase Kit (KIT) KIT_HUMAN Inhibitor REF00003966 DG01624 Tyrosine-protein kinase Kit (KIT) KIT_HUMAN Inhibitor REF00004392 DG01637 Tyrosine-protein kinase Mer (MERTK) MERTK_HUMAN Inhibitor REF00003917 DG01638 Tyrosine-protein kinase Mer (MERTK) MERTK_HUMAN Inhibitor REF00003918 DG01640 Tyrosine-protein kinase Mer (MERTK) MERTK_HUMAN Inhibitor REF00004375 DG01267 Tyrosine-protein kinase UFO (AXL) UFO_HUMAN . REF00003076 DG01902 Ubiquitin-protein ligase E3 Mdm2 (MDM2) MDM2_HUMAN Antagonist REF00004574 DG00620 Urokinase plasminogen activator surface receptor (PLAUR) UPAR_HUMAN Inhibitor REF00003699 DG01550 Urokinase plasminogen activator surface receptor (PLAUR) UPAR_HUMAN Inhibitor REF00004461 DG00662 Varicella-zoster virus DNA polymerase (VZV ORF28) DPOL_VZVD Modulator REF00003354 DG00402 Vascular endothelial growth factor A (VEGFA) VEGFA_HUMAN Inhibitor REF00000712 DG00650 Vascular endothelial growth factor A (VEGFA) VEGFA_HUMAN Inhibitor REF00003672 DG00651 Vascular endothelial growth factor A (VEGFA) VEGFA_HUMAN Inhibitor REF00003792 DG00128 Vascular endothelial growth factor receptor (VEGFR) . Modulator REF00001742 DG00244 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00001374 DG00250 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Modulator REF00002753 DG00282 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Modulator REF00002738 DG00332 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00002310 DG00617 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00003330 DG00619 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00003376 DG01166 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00003682 DG01260 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00003230 DG01521 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00004260 DG01522 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00003966 DG01599 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Antagonist REF00004377 DG01802 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Inhibitor REF00004070 DG01892 Vascular endothelial growth factor receptor 2 (KDR) VGFR2_HUMAN Modulator REF00004592 DG01126 Vasopressin receptor (VR) NOUNIPROTAC Agonist REF00003820 DG01489 Vasopressin receptor (VR) NOUNIPROTAC Agonist REF00004539 DG01007 Vasopressin V1a receptor (V1AR) V1AR_HUMAN Inhibitor REF00003756 DG01126 Vasopressin V1a receptor (V1AR) V1AR_HUMAN Inhibitor REF00003820 DG01489 Vasopressin V1a receptor (V1AR) V1AR_HUMAN Inhibitor REF00004539 DG01126 Vasopressin V1b receptor (V1BR) V1BR_HUMAN Antagonist REF00003820 DG01489 Vasopressin V1b receptor (V1BR) V1BR_HUMAN Antagonist REF00004539 DG01007 Vasopressin V2 receptor (V2R) V2R_HUMAN Antagonist REF00003756 DG01059 Vasopressin V2 receptor (V2R) V2R_HUMAN Antagonist REF00003250 DG01126 Vasopressin V2 receptor (V2R) V2R_HUMAN Antagonist REF00003820 DG01489 Vasopressin V2 receptor (V2R) V2R_HUMAN Antagonist REF00004539 DG01606 V-erbA-related protein 1 (NR1D1) NR1D1_HUMAN Antagonist REF00004474 DG01607 V-erbA-related protein 1 (NR1D1) NR1D1_HUMAN Antagonist REF00004387 DG00268 Vitamin D3 receptor (VDR) VDR_HUMAN Agonist REF00002059 DG00249 Voltage-gated calcium channel alpha Cav3.1 (CACNA1G) CAC1G_HUMAN Blocker REF00002865 DG00902 Voltage-gated calcium channel alpha Cav3.1 (CACNA1G) CAC1G_HUMAN Blocker (channel blocker) REF00003267 DG01074 Voltage-gated L-type calcium channel (L-CaC) NOUNIPROTAC Blocker REF00003401 DG00014 Voltage-gated potassium channel Kv11.1 (KCNH2) KCNH2_HUMAN Activator REF00002651 DG00799 Voltage-gated sodium channel (Nav) NOUNIPROTAC Modulator REF00003219 DG01223 Voltage-gated sodium channel (Nav) NOUNIPROTAC Modulator REF00003740 DG00269 Voltage-gated sodium channel alpha Nav1.8 (SCN10A) SCNAA_HUMAN Inhibitor REF00001267 DG00824 Voltage-gated sodium channel alpha Nav1.8 (SCN10A) SCNAA_HUMAN Blocker REF00003008 DG01781 Voltage-gated sodium channel alpha Nav1.8 (SCN10A) SCNAA_HUMAN Blocker REF00004336 DG00592 Voltage-gated sodium channel alpha Nav1.9 (SCN11A) SCNBA_HUMAN Blocker REF00003317 DG00623 Voltage-gated sodium channel alpha Nav1.9 (SCN11A) SCNBA_HUMAN Blocker REF00003593 DG00639 Voltage-gated sodium channel alpha Nav1.9 (SCN11A) SCNBA_HUMAN Blocker REF00003593 DG00750 Voltage-gated sodium channel alpha Nav1.9 (SCN11A) SCNBA_HUMAN Blocker REF00003192 DG00546 Wee1-like protein kinase (WEE1) WEE1_HUMAN Inhibitor REF00003670 DG00010 Xanthine dehydrogenase/oxidase (XDH) XDH_HUMAN Inhibitor REF00002302 DG00103 Xanthine dehydrogenase/oxidase (XDH) XDH_HUMAN Inhibitor REF00002220 DG01003 Xanthine dehydrogenase/oxidase (XDH) XDH_HUMAN Inhibitor REF00003703 DG01312 Xanthine dehydrogenase/oxidase (XDH) XDH_HUMAN Inhibitor REF00003127